Nano-aperture 30-element triphenylamine rigid macrocyclic compound and preparation method thereof
A technology of macrocyclic compounds and triphenylamine, which is applied in the direction of organic chemistry, can solve the problems of low conversion rate, can not be used as high carrier mobility material, etc., and achieve high total conversion rate, low cost and easy availability of raw materials Effect
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Embodiment 1
[0046] Synthesis of 4-methyl-N-phenylaniline
[0047] In a 100mL single-necked flask, add 30mmol iodobenzene, 33mmol p-toluidine, 3mmol cuprous iodide, 6mmol L-proline, 60mmol K 2 CO 3 and 80 mL of DMSO. Under the protection of nitrogen, stir and heat to 110°C, keep the temperature for 24 hours; cool down to room temperature, add cold 2N hydrochloric acid to make the pH value reach 7, filter into a 250mL separatory funnel, extract three times with 50mL ethyl acetate each time, The organic phase was washed with saturated brine, then dried by adding anhydrous sodium sulfate, the solvent was removed under vacuum, and separated by column chromatography to obtain white floc 4-methyl-N-phenylaniline with a conversion rate of 45%.
[0048] The reaction equation is as follows:
[0049]
Embodiment 2
[0051] Synthesis of 4-bromo-N-phenyl-N-p-methylaniline
[0052] In a 100mL one-necked flask, add 18mmol p-bromoiodobenzene, 15mmol 4-methyl N-phenylaniline, 1.5mmol cuprous iodide, 3mmol L-proline, 30mmol K 2 CO 3 and 80 mL of DMSO. Under the protection of nitrogen, stir and heat to 110°C, keep the temperature for 24 hours; cool down to room temperature, add 2N hydrochloric acid to make the pH value reach 7, filter into a 250mL separatory funnel, extract three times with 25mL ethyl acetate each time, organic phase Wash with saturated brine, then add anhydrous sodium sulfate to dry; remove the solvent under vacuum, and separate through chromatography column to obtain white wax 4-bromo-N-phenyl-N-p-methylaniline, the conversion rate is 75%.
[0053] The reaction equation is as follows:
[0054]
Embodiment 3
[0056] Synthesis of 4-bromo-N-(4-bromophenyl)-N-phenylaniline
[0057] In a 100mL single-necked flask, add 30mmol aniline, 72mmol p-toluidine, 3mmol cuprous iodide, 6mmol L-proline, 60mmol K 2 CO 3 and 80mL of DMSO, under nitrogen protection, stirred, heated to 110°C, and kept at a constant temperature for 24 hours; lowered to room temperature, added 2N hydrochloric acid to make the pH value reach 7, filtered into a 250mL separatory funnel, each time with 50mL ethyl acetate Extracted three times, the organic phase was washed with saturated brine, and then dried by adding anhydrous sodium sulfate; the solvent was removed under vacuum; after separation by chromatography column, a white waxy substance, 4-bromo-N-(4-bromophenyl) -N-phenylaniline, the conversion rate was 88%.
[0058] The reaction equation is as follows:
[0059]
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