Asymmetric bis-quaternary ammonium salt as well as preparation method and application thereof
A double quaternary ammonium salt, asymmetric technology, applied in the field of quaternary ammonium salt fungicides, can solve the problems of complex process steps, low yield, long synthesis time and the like
- Summary
- Abstract
- Description
- Claims
- Application Information
AI Technical Summary
Problems solved by technology
Method used
Image
Examples
preparation example Construction
[0165] The preparation method of unsymmetrical double quaternary ammonium salt of the present invention:
[0166] 1. Weigh raw materials by molar ratio: compound 2 (secondary amine): compound 1 (saturated monohalogenated hydrocarbon): compound 3 (epoxyhalopropane): compound 4 (R 4 , R 5 , R 6 Substituted tertiary amine)=0.9~1.1: 0.8~1.7: 0.8~1.5: 0.5~1.4;
[0167] 2. Add additives of 0.8-6% of the total weight of raw materials and catalysts of 0.3-3% of the total weight of raw materials, mix well and react at 40-100°C for 0.8-1.7h, then react at 90-150°C for 1.8-2.7h have to.
[0168] The catalyst is an amide compound, such as N, N-R 7 , R 8 Replace -R 9 Substituted amides, R 7 , R 8 , R 9 are independently H or C1-C8 alkyl.
[0169] The catalyst is preferably at least one of formamide, N,N-dimethylformamide, N,N-dimethylacetamide, and N,N-diethylformamide.
[0170] The auxiliary agent is an alkyl alcohol with 8 carbons or less, preferably at least one of ethanol, n...
Embodiment 1
[0181] Example 1: Weigh the raw materials according to the molar ratio of benzyl chloride: epichlorohydrin: dodeca / tetradecylamine: diethylamine is 1.2:0.9:0.8:1. The amount of auxiliary alcohols is 3% of the total weight of the raw materials, and the amount of the catalyst amide is 1.0% of the total weight of the raw materials. Put the above materials in the reactor, turn on the stirrer to heat, control the reaction temperature at 60-100°C, after 1.5h of reaction, turn on the heating device, raise the temperature to 100°C, and control the reaction temperature at 100-140°C, and react for 2.5h , cooled to about 90°C and discharged. The appearance is a reddish-brown viscous liquid, the content of the active substance is 93.5% and the yield is 94.8% according to the analysis method of the quaternary ammonium salt.
[0182] Analysis and detection method of quaternary ammonium salt: quaternary ammonium salt is a cationic surfactant, which can form a chelate with dichlorofluorescen...
Embodiment 2
[0183] Example 2: The raw materials were weighed according to the molar ratio of ethyl bromide: epichlorohydrin: hexadecyl / octadecyl tertiary amine: diphenylamine 1.4: 1.0: 0.8: 1. Auxiliary alcohols are 2% of the total dosage, catalyst amides are 0.5% of the total dosage, and the above materials are placed in the reactor. Turn on the stirrer to heat, control the reaction temperature at 60-100°C, after 1.5 hours of reaction, turn on the heating device, raise the temperature to 100°C, and control the reaction temperature to 100-140°C, react for 2.0 hours, cool to about 90°C and discharge. The appearance is a reddish-brown viscous liquid, and its active matter content is 94.1% and the yield is 93.8% as determined by referring to the analysis method of quaternary ammonium salt.
PUM
Login to View More Abstract
Description
Claims
Application Information
Login to View More 


