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Preparation method and application of targeting chondrocyte drug delivery system

A chondrocyte and delivery system technology, applied in the fields of genetic engineering and biomedicine, can solve the problem of low therapeutic potential of cell-targeted delivery of drug molecules, and achieve the effects of controlling the destruction of articular cartilage, promoting cartilage repair, and slowing down degradation.

Inactive Publication Date: 2021-08-24
THE SECOND PEOPLES HOSPITAL OF SHENZHEN
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  • Summary
  • Abstract
  • Description
  • Claims
  • Application Information

AI Technical Summary

Problems solved by technology

[0003] The present invention designs the preparation method and application of the drug delivery system targeting chondrocytes to solve the disadvantages of low therapeutic potential of cell-targeted delivery drug molecules

Method used

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Examples

Experimental program
Comparison scheme
Effect test

Embodiment 1

[0025] The present invention provides a technical solution: a preparation method and application of a chondrocyte-targeted drug delivery system, the method comprising the following steps:

[0026] S1: Construct a plasmid, and use the chondrocyte-carrying affinity peptide (CAP) to be fused and expressed on the exosome membrane protein (lamp2b) as a targeted genetically engineered exosome that can target chondrocytes;

[0027] S2: Screen stable cell lines, express plasmid CAP-lamp2b in DC cells, and screen stable cell lines;

[0028] S3: Extract cartilage-affinity-targeted exosomes, use exosome-free medium to expand cells stably expressing CAP-lamp2b, collect cell supernatant, and perform differential ultracentrifugation to obtain exosomes. 1. Design of lamp2b Primer, using mouse cDNA as a template, PCR amplification obtains the lamp2b fragment, PCR (polymerase chain reaction) purification;

[0029] 2. Cloning the lamp2b gene after step 1 PCR purification and recovery into the ...

Embodiment 2

[0040] The present invention provides a technical solution: a preparation method and application of a chondrocyte-targeted drug delivery system, the method comprising the following steps:

[0041] S1: Construct a plasmid, and use the chondrocyte-carrying affinity peptide (CAP) to be fused and expressed on the exosome membrane protein (lamp2b) as a targeted genetically engineered exosome that can target chondrocytes;

[0042] S2: Screen stable cell lines, express plasmid CAP-lamp2b in DC cells, and screen stable cell lines;

[0043] S3: Extract cartilage-affinity-targeted exosomes, use exosome-free medium to expand cells stably expressing CAP-lamp2b, collect cell supernatant, and perform differential ultracentrifugation to obtain exosomes. 1. Design of lamp2b Primer, using mouse cDNA as a template, PCR amplification obtains the lamp2b fragment, PCR (polymerase chain reaction) purification;

[0044] 2. Cloning the lamp2b gene after step 1 PCR purification and recovery into the ...

Embodiment 3

[0055] The present invention provides a technical solution: a preparation method and application of a chondrocyte-targeted drug delivery system, the method comprising the following steps:

[0056] S1: Construct a plasmid, and use the chondrocyte-carrying affinity peptide (CAP) to be fused and expressed on the exosome membrane protein (lamp2b) as a targeted genetically engineered exosome that can target chondrocytes;

[0057] S2: Screen stable cell lines, express plasmid CAP-lamp2b in DC cells, and screen stable cell lines;

[0058] S3: Extract cartilage-affinity-targeted exosomes, use exosome-free medium to expand cells stably expressing CAP-lamp2b, collect cell supernatant, and perform differential ultracentrifugation to obtain exosomes. 1. Design of lamp2b Primer, using mouse cDNA as a template, PCR amplification obtains the lamp2b fragment, PCR (polymerase chain reaction) purification;

[0059] 2. Cloning the lamp2b gene after step 1 PCR purification and recovery into the ...

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Abstract

The invention relates to the field of genetic engineering and biomedicine, and discloses a preparation method and application of a targeted chondrocyte drug delivery system, and the method comprises the following steps: S1, constructing plasmids; S2, screening stable cell strains; S3, extracting a cartilage affinity targeting exosome; S4, loading an exogenous miRNA-140; S5, carrying out targeted delivery on the miRNA-140. According to the invention, the treatment potential of the miRNA medicine is realized, and the efficient tissue-specific delivery medicine is used for treating osteoarthritis. According to the invention, exosome surface mask protein lamp2b is subjected to genetic engineering modification, and cartilage cell affinity peptide is fused with exosome surface mask protein lamp2b, so that exosome can target specific soft cells, and miRNA drug molecules are carried to treat various osteoarthritis.

Description

technical field [0001] The invention relates to the fields of genetic engineering and biomedicine, in particular to a preparation method and application of a drug delivery system targeting chondrocytes. Background technique [0002] Targeted delivery of drug molecules to specific cell types is a major challenge in precision medicine. Natural exosomes have biologically functionalized nanovesicles, which can display a variety of ligands targeting proteins or polypeptides through genetic engineering and directly package drugs to exercise targeted drug delivery capabilities. [0003] The present invention designs a preparation method and application of a targeted chondrocyte drug delivery system to solve the disadvantage of low therapeutic potential of cell-targeted drug delivery. Contents of the invention [0004] The purpose of the present invention is to provide a preparation method and application of a chondrocyte-targeted drug delivery system, so as to solve the problems...

Claims

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Application Information

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Patent Type & Authority Applications(China)
IPC IPC(8): C12N15/85C12N15/62C12N5/10A61K47/46A61K47/42A61K31/7105A61P19/02A61P19/08A61P29/00
CPCA61K9/0019A61K31/7105A61K47/42A61K47/46A61P19/02A61P19/08A61P29/00C07K14/47C07K2319/33C12N5/0639C12N15/111C12N15/85C12N2320/32C12N2509/00C12N2510/00C12N2800/107
Inventor 梁宇杰徐丽梅段莉徐晓
Owner THE SECOND PEOPLES HOSPITAL OF SHENZHEN