Dosing of cabozantinib formulations

MA39735AUndetermined Publication Date: 2017-01-25EXELIXIS INC
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Patent Information

Application Number
MA39735
Authority / Receiving Office
MA · MA
Patent Type
Applications
Current Assignee / Owner
Priority Date
2014-03-17
Filing Date
2015-03-17
Publication Date
2017-01-25
Patent Text Reader

Abstract

The invention relates to administration of various pharmaceutical formulations of n- (4-{[6,7-bis(methyloxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1- dicarboxamide, (cabozantinib) a c-met inhibitor, and its metabolites, to achieve desirable pharmacokinetic and pharmacodynamic effects.
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