Methods of identifying patients likely to benefit from treatment with a telomerase inhibitor
Patent Information
- Application Number
- IL279623
- Authority / Receiving Office
- IL · IL
- Patent Type
- Applications
- Current Assignee / Owner
- Priority Date
- 2018-11-29
- Filing Date
- 2019-07-29
- Publication Date
- 2026-07-01
- Estimated Expiration
- 2039-07-29
AI Technical Summary
Current treatments for myelofibrosis, particularly those lacking mutations in JAK2, CALR, and MPL genes or having high-molecular risk mutations in ASXL1, EZH2, SRSF2, and IDH1/2, do not effectively address the disease progression and survival outcomes for patients, as they often lead to leukemic transformation and shortened overall survival.
Identifying patients with triple negative status or high-molecular risk based on genetic mutations using DNA samples from bone marrow or peripheral blood, and administering a telomerase inhibitor like imetelstat to target and inhibit telomerase activity, thereby potentially slowing disease progression.
The approach effectively identifies patients likely to benefit from telomerase inhibitor treatment, leading to improved spleen volume reduction, symptom response, and overall survival, particularly in patients with triple negative or high-molecular risk profiles, offering a new therapeutic option for myelofibrosis management.