Pharmaceutically acceptable salts, crystalline forms, and uses of diaminocyclopentyl-substituted heteroaryl derivatives

TW202635678APending Publication Date: 2026-09-01JIANGSU HENGRUI MEDICINE CO LTD
View PDF 0 Cites 0 Cited by

Patent Information

Application Number
TW115102672
Authority / Receiving Office
TW · TW
Patent Type
Applications
Current Assignee / Owner
Priority Date
2025-01-23
Filing Date
2026-01-22
Publication Date
2026-09-01

Smart Images

  • Figure TWG2TA001075194_001
    Figure TWG2TA001075194_001
  • Figure TWG2TA001075194_002
    Figure TWG2TA001075194_002
  • Figure TWG2TA001075194_003
    Figure TWG2TA001075194_003
Patent Text Reader

Abstract

The present disclosure relates to pharmaceutically acceptable salts, crystalline forms, and uses of diaminocyclopentyl-substituted heteroaryl derivatives. Specifically, the present disclosure provides pharmaceutically acceptable salts, crystal forms, and preparation methods of 1-(6-{[(1S,3S)-3-(6,7-dihydro[1,4]dioxepino[3,2-d]pyrimidin-2-ylamino)cyclopentyl]amino}pyridin-3-yl)-1,2-dihydropyridin-2-one, which exhibit excellent stability and are suitable for clinical applications.
Need to check novelty before this filing date? Find Prior Art