Ad5 E1-E2b- Viral Vector for Repeated Immunotherapy

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Solution Overview

Problem

First-generation adenovirus vector vaccines, such as Ad5 [E1-] vectors, face limitations due to pre-existing anti-adenovirus neutralizing antibodies and immune responses, leading to inadequate immune stimulation and adverse effects, particularly in individuals with prior adenovirus exposure, limiting their use for repeated vaccinations and cancer immunotherapy.

Innovation Solution

Development of second-generation adenovirus vectors with deletions in the E1 and E2b regions, specifically Ad5 [E1-, E2b-] vectors, which reduce late phase viral protein expression, minimize immune responses to viral proteins, and allow for multiple vaccinations by inducing potent antigen-specific immune responses even in immune-hosts, while maintaining safety and efficacy.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Power

If first-generation Ad5 vectors are used for vaccination, then robust T-cell-mediated immune responses can be induced, but pre-existing anti-Ad5 neutralizing antibodies and immune responses eliminate the vector and transduced cells, limiting repeated vaccinations

Engineering Contradiction:
Improveimmune response induction capabilityVSAvoidrepeated vaccination capability
Core Design Contradiction:
PowerVSReliability

Solution Approach 1:

The patent extracts and removes the E2b gene region from the adenovirus vector, which encodes viral proteins that trigger strong immune responses. By deleting this region, the vector maintains its ability to deliver therapeutic genes while reducing immunogenicity, allowing repeated administrations without being eliminated by pre-existing immunity

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent modifies the viral vector by deleting the E2b gene region, fundamentally changing the vector's properties. This genetic modification reduces the expression of viral proteins that trigger immune responses, transforming the vector from one that is rapidly eliminated to one that can sustain long-term transgene expression and withstand repeated administrations

Inventive Principle:
Principle #35Parameter changes

2Reliability

If adenovirus vectors are used to deliver tumor-associated antigens, then cancer immunotherapy survival benefits can be achieved, but host immune responses eliminate the vector and virally transduced cells, reducing sustained long-term expression

Engineering Contradiction:
Improvecancer immunotherapy efficacyVSAvoidtransgene expression duration
Core Design Contradiction:
ReliabilityVSDuration of action of stationary object

Solution Approach 1:

By extracting and removing the E2b gene region from the adenovirus vector, the patent reduces the expression of viral proteins that are targets of host immune responses. This allows the vector to evade immune detection and elimination, enabling sustained long-term transgene expression necessary for effective cancer immunotherapy

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent applies partial deletion of the adenovirus genome (specifically the E2b region) rather than complete removal. This partial modification is sufficient to reduce immunogenicity and enable long-term expression while maintaining the vector's essential functions for gene delivery and immune response induction against tumor antigens

Inventive Principle:
Principle #16Partial or excessive action

3Power

If vaccine doses are increased to overcome pre-existing immunity and induce desired CMI responses, then immune response can be enhanced, but unacceptable adverse effects result

Engineering Contradiction:
Improvecell-mediated immunity responseVSAvoidadverse effects
Core Design Contradiction:
PowerVSObject-affected harmful factors

Solution Approach 1:

The patent changes the immunogenicity parameter of the vector by deleting the E2b gene region. This modification allows the vector to induce desired cell-mediated immunity responses at lower, safer doses by reducing the immune response against viral proteins themselves, thereby separating the therapeutic immune response from the harmful adverse effects

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3242940B1Methods and compositions for combination immunotherapy
Publication Date: 2023.03.29 ETUBICS CORP
  • EP3242940B1 patent drawingFigure 1~2
  • EP3242940B1 patent drawingFigure 3
  • EP3242940B1 patent drawingFigure 4A~4B

AI summary

Methods for generating immune responses using adenovirus vectors that allow multiple vaccinations with the same adenovirus vector and vaccinations in individuals with preexisting immunity to adenovirus are provided.