Amorphous Solid Cannabis Aerosol Composition

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Solution Overview

Problem

Current methods for delivering cannabis constituents, such as CBD, in aerosol form face limitations due to solubility issues in liquid vaping systems, leading to suboptimal delivery of high levels of these compounds.

Innovation Solution

An amorphous solid composition comprising 1-50 wt% cannabis constituents, 10-80 wt% aerosol-former materials like glycerol, and gelling agents including cellulose derivatives, which forms a monolithic solid capable of generating aerosols when heated, allowing for higher delivery of cannabis compounds.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Quantity of substance

If liquid vaping systems are used to deliver cannabis constituents, then the delivery mechanism is simple, but the solubility of cannabis compounds is limited

Engineering Contradiction:
Improveconcentration of cannabis compoundsVSAvoidsolubility in liquid medium
Core Design Contradiction:
Quantity of substanceVSReliability

Solution Approach 1:

The patent changes the physical state of the cannabis compound delivery system from liquid to amorphous solid. This parameter change allows cannabis constituents to be delivered at higher concentrations (1-50 wt%) without solubility limitations, as the amorphous solid matrix does not require dissolution in a liquid medium to release the active compounds during heating.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite amorphous solid material comprising cannabis constituents combined with aerosol-forming materials and gelling agents. This composite structure enables the integration of multiple functions: the cannabis provides the active compound, the aerosol-forming materials enable vaporization, and the gelling agents provide structural stability, collectively resolving the solubility limitation while maintaining reliable delivery.

Inventive Principle:
Principle #40Composite materials

2Quantity of substance

If high levels of cannabis compounds are delivered, then the therapeutic effect is improved, but the solubility limitations in liquid systems prevent effective delivery

Engineering Contradiction:
Improveamount of cannabis compounds deliveredVSAvoidformulation stability
Core Design Contradiction:
Quantity of substanceVSEase of manufacture

Solution Approach 1:

By transitioning from liquid to amorphous solid formulation, the patent enables incorporation of high levels of cannabis compounds (1-50 wt%) without the solubility constraints that limit liquid systems. The amorphous solid state provides a stable matrix that maintains formulation integrity while allowing high active compound loading.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent introduces gelling agents as intermediary materials that stabilize the amorphous solid structure containing high concentrations of cannabis compounds. These gelling agents act as a mediating matrix that maintains formulation stability while enabling high levels of active compound incorporation, resolving the conflict between quantity and manufacturability.

Inventive Principle:
Principle #24Intermediary (Mediator)

3Quantity of substance

If amorphous solid composition is used, then higher cannabis compound delivery is achieved, but the manufacturing process becomes more complex

Engineering Contradiction:
Improveconcentration of cannabis compoundsVSAvoidcomposition structure
Core Design Contradiction:
Quantity of substanceVSDevice complexity

Solution Approach 1:

The patent employs composite materials comprising cannabis constituents, aerosol-forming materials, and gelling agents in an amorphous solid matrix. This composite approach enables high cannabis compound concentration (1-50 wt%) while the combination of components works synergistically to simplify the overall formulation process compared to attempting to dissolve high concentrations in liquid systems.

Inventive Principle:
Principle #40Composite materials

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The amorphous solid composition enables the efficient delivery of higher cannabis compound levels by forming a monolithic solid that aerosolizes effectively when heated, overcoming solubility limitations in traditional vaping systems.

Implementation Method 1

The amorphous solid composition enables the efficient delivery of higher cannabis compound levels by forming a monolithic solid that aerosolizes effectively when heated

Methodology Applied
Scientific EffectVaporization: Evaporation

Implementation Method 2

gelling agent, the gelling agent comprising cellulose or a derivative thereof, and a non-cellulosic gelling agent

Methodology Applied
Scientific EffectGel formation: Gel

Data Source

PatentEP4208046B1Compositions and methods
Publication Date: 2024.11.06 NICOVENTURES TRADING LTD
  • EP4208046B1 patent drawingFigure 1~2
  • EP4208046B1 patent drawingFigure 3~4
  • EP4208046B1 patent drawingFigure 5

AI summary

The present invention provides an amorphous solid for use in aerosol generation, the amorphous solid comprising: about 1 to about 50 wt% constituent, derivative or extract of cannabis; about 10 to about 80 wt% aerosol-former material; gelling agent, the gelling agent comprising cellulose or a derivative thereof, and a non-cellulosic gelling agent; and optionally filler, wherein the amount of gelling agent and optional filler taken together is from about 10 to about 60 wt%; wherein the wt% values are calculated on a dry weight basis.