Anilide Herbicide Suspension Stability via Anionic Surfactant

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Solution Overview

Problem

Formulating stable, water-based suspension concentrates of sparingly soluble anilide herbicides is challenging due to Ostwald ripening, which leads to particle size growth, crystal formation, and instability, affecting shelf-life and application efficacy.

Innovation Solution

A stable agrochemical composition comprising a dispersed phase of pre-treated anilide herbicide and a continuous aqueous phase with at least one anionic surfactant, where the anilide herbicide is pre-treated through heat processes to stabilize the molecule, and the composition is formulated as a suspension concentrate with controlled particle size distribution.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Ease of manufacture

If anilide herbicide is formulated as aqueous suspension concentrate, then water-based dispersion is achieved, but Ostwald ripening causes particle size growth and crystal formation

Engineering Contradiction:
Improvewater-based dispersionVSAvoidparticle size stability
Core Design Contradiction:
Ease of manufactureVSStability of the object's composition

Solution Approach 1:

The patent introduces a specific dispersant as an intermediary substance between the anilide herbicide particles and water. This dispersant adsorbs onto the particle surfaces, providing steric or electrostatic repulsion that prevents particle aggregation and Ostwald ripening, thereby maintaining stable particle size distribution in the aqueous suspension concentrate.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent modifies the surface properties of anilide herbicide particles through treatment with specific dispersants, changing parameters such as surface charge, hydrophilicity, and surface energy. These parameter changes prevent particle aggregation and crystal growth, enabling stable water-based formulations without Ostwald ripening.

Inventive Principle:
Principle #35Parameter changes

2Ease of manufacture

If conventional surfactants are used to facilitate dispersion, then dispersion is improved, but solubility modification leads to aqueous phase instability

Engineering Contradiction:
Improvedispersion facilitationVSAvoidaqueous phase stability
Core Design Contradiction:
Ease of manufactureVSStability of the object's composition

Solution Approach 1:

The patent employs specific dispersants that function effectively at low concentrations and provide stable dispersion without long-term solubility issues. These dispersants are selected to provide sufficient stabilization during the product shelf life without causing delayed solubility changes or phase separation.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The dispersant acts as an intermediary that facilitates particle-water interaction without significantly altering the solubility equilibrium of the anilide herbicide. This prevents the harmful effect of modified solubility while achieving good dispersion.

Inventive Principle:
Principle #24Intermediary (Mediator)

3Object-affected harmful factors

If particles are suspended in aqueous medium, then inhalation danger is reduced, but particle settling occurs during storage

Engineering Contradiction:
Improveinhalation risk reductionVSAvoidparticle suspension stability
Core Design Contradiction:
Object-affected harmful factorsVSStability of the object's composition

Solution Approach 1:

The dispersant serves as an intermediary that provides repulsive forces between particles, counteracting gravitational settling. This creates a kinetically stable suspension where particles remain dispersed during storage, eliminating both inhalation risks and settling problems.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent creates a dynamic equilibrium in the suspension where repulsive forces from the dispersant continuously counteract gravitational attraction, preventing particle settling while maintaining safe water-based formulation for reduced inhalation exposure.

Inventive Principle:
Principle #15Dynamics

Data Source

PatentUS11751565B2Stable agrochemical composition
Publication Date: 2023.09.12 UPL CORPORATION LTD(MU)

AI summary

The present invention provides a stable agrochemical composition including a dispersed phase comprising an anilide herbicide; a continuous aqueous phase; and at least one anionic surfactant. The present invention also provides a process of preparing stable agrochemical compositions and methods of application thereof.