Antigen-MHC Nanoparticle Complexes for MS Tolerance

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Solution Overview

Problem

Current therapies for multiple sclerosis (MS) are often poorly tolerated and have significant side effects, with a need for more effective and better-tolerated treatments that can manage the disease effectively without compromising systemic immunity.

Innovation Solution

Administration of antigen-MHC-nanoparticle complexes, specifically designed to expand anti-pathogenic autoreactive T-cells, which are biocompatible and bioabsorbable, to treat or prevent MS by targeting multiple sclerosis-related antigens, thereby reducing disease severity and inflammation.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If conventional MS medications are used, then MS attacks can be eased and disease progression can be slowed, but significant side effects and poor tolerance occur

Engineering Contradiction:
Improvedisease management effectivenessVSAvoidside effects and tolerance
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent uses nanoparticle complexes as intermediary carriers that deliver antigen-MHC complexes to T-cells. These nanoparticles serve as a mediator between the therapeutic agent and the immune system, enabling targeted delivery while minimizing off-target effects and improving tolerance compared to conventional medications.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The invention applies local quality by targeting specific T-cell populations with antigen-MHC-nanoparticle complexes in a localized manner. The therapy is designed to act specifically on pathogenic T-cells while preserving overall immune function, thereby reducing system-wide side effects while maintaining therapeutic effectiveness in the CNS.

Inventive Principle:
Principle #3Local quality

2Reliability

If therapies are developed to expand anti-pathogenic autoreactive T-cells, then MS symptoms can be reduced, but the complexity of the treatment protocol increases

Engineering Contradiction:
Improvesymptom reductionVSAvoidtreatment protocol complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent merges multiple functions into a single nanoparticle complex: the nanoparticle serves as both the delivery vehicle and the presentation platform for antigen-MHC complexes. This consolidation simplifies the treatment protocol by eliminating the need for separate administration of multiple agents, while still achieving the goal of expanding anti-pathogenic T-cells.

Inventive Principle:
Principle #5Merging (Combining)

3Reliability

If apoptosis-inducing molecules are used for tolerance induction, then antigen-specific tolerance can be achieved, but significant side effects occur

Engineering Contradiction:
Improveantigen-specific toleranceVSAvoidside effects
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent converts the potentially harmful effect of apoptosis-inducing molecules into a beneficial tolerance induction mechanism. By using nanoparticle-delivered antigen-MHC complexes to activate regulatory T-cells, the therapy achieves antigen-specific tolerance without the severe side effects associated with direct apoptosis induction, effectively turning a harmful mechanism into a beneficial therapeutic approach.

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Data Source

PatentEP2906594B1Methods and compositions for treating multiple sclerosis and related disorders
Publication Date: 2018.12.05 UTI LIMITED PARTNERSHIP
  • EP2906594B1 patent drawingFigure 1
  • EP2906594B1 patent drawingFigure 2
  • EP2906594B1 patent drawingFigure 3

AI summary

This disclosure provides therapeutic compositions and methods for treating multiple sclerosis or a multiple sclerosis-related disorder in a subject in need thereof comprising administering an effective amount of an antigen-MHC-nanoparticle complex to the subject, wherein the antigen is a multiple sclerosis-related antigen.