BAFF Polypeptide for Selective Plasma Cell Targeting in Multiple Sclerosis

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Solution Overview

Problem

Current treatments for autoimmune diseases like multiple sclerosis, such as anti-CD20 therapy and atacicept, do not effectively target plasma cells and can lead to disease exacerbations, highlighting a need for improved methods to regulate B cells and reduce inflammation in autoimmune diseases.

Innovation Solution

A composition comprising a B-cell Activating Factor (BAFF) polypeptide, an agent that promotes the survival and migration of gut-derived commensal-reactive B cells to the central nervous system, or an agent that depletes B cells, or a gut commensal that increases IgA levels, to treat autoimmune diseases by enriching gut-derived commensal-reactive IgA+ plasmablasts and plasma cells in the central nervous system.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If anti-CD20 therapy is used to deplete B cells, then B cell depletion is achieved, but plasma cells are not effectively targeted and disease exacerbations occur

Engineering Contradiction:
Improveeffectiveness of B cell targetingVSAvoiddisease exacerbation
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

Instead of depleting all B cells (including protective ones), the invention inverts the approach by selectively depleting only pathogenic plasma cells through anti-CD38 therapy, while preserving regulatory B cells that produce IgA and IL-10. This selective inversion resolves the contradiction by achieving reliable pathogen targeting without causing disease exacerbation.

Inventive Principle:
Principle #13The other way round (Inversion)

Solution Approach 2:

The invention applies local quality by differentiating between various B cell subsets and targeting only the pathogenic plasma cells with anti-CD38 therapy. By distinguishing pathogenic from protective B cells and applying selective depletion, the therapy achieves reliable pathogen targeting while avoiding harm to regulatory B cells.

Inventive Principle:
Principle #3Local quality

2Object-affected harmful factors

If B cells are depleted to reduce inflammation, then inflammatory responses are suppressed, but immunoregulatory functions are also lost

Engineering Contradiction:
ImproveinflammationVSAvoidimmunoregulatory function
Core Design Contradiction:
Object-affected harmful factorsVSReliability

Solution Approach 1:

The invention inverts the conventional approach by not depleting regulatory B cells but instead enhancing their function. By using agents that promote the survival and migration of regulatory IgA+ plasma cells and by depleting only pathogenic cells, the therapy reduces inflammation while maintaining or enhancing immunoregulatory functions.

Inventive Principle:
Principle #13The other way round (Inversion)

Solution Approach 2:

The invention applies local quality by selectively targeting pathogenic B cells while preserving and enhancing regulatory B cell functions. Through selective depletion and promotion of specific B cell subsets, the therapy achieves inflammation reduction without compromising immunoregulatory reliability.

Inventive Principle:
Principle #3Local quality

3Ease of manufacture

If conventional therapies are used to treat autoimmune diseases, then treatment is provided, but plasma cells are not effectively targeted

Engineering Contradiction:
Improvetreatment availabilityVSAvoidplasma cell targeting
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The invention changes the targeting parameter from CD20 (conventional therapy) to CD38 (pathogenic plasma cells). By using anti-CD38 therapy and selective agents that target plasma cells based on their specific markers and functions, the invention achieves reliable plasma cell targeting while maintaining treatment availability.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3883593B1BAFF polypeptide for use in treating multiple sclerosis
Publication Date: 2024.03.06 F HOFFMANN LA ROCHE LTD
  • EP3883593B1 patent drawingFigure 1a~1f
  • EP3883593B1 patent drawingFigure 2A~2F
  • EP3883593B1 patent drawingFigure 3a~3h

AI summary

The present disclosure provides methods of treating an autoimmune disease (e.g., multiple sclerosis) or reducing inflammation by administering at least a B-cell activating Factor (BAFF) polypeptide to a subject in need thereof. The effect of BAFF on plasmablast/plasma cells and their role in autoimmune diseases is also disclosed.