Beraprost Adjuvant Mitigates CAR T-Cell Cytokine Release Syndrome

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Solution Overview

Problem

CAR T-cell therapies are effective but suffer from significant side effects such as cytokine release syndrome (CRS), which affects a high percentage of patients and can be fatal, necessitating the development of new treatments to reduce or eliminate these undesired effects.

Innovation Solution

Administering CAR T-cells in conjunction with a pharmaceutical composition containing prostacyclin/prostaglandin analogs, such as beraprost, to mitigate CRS symptoms by reducing cytokine production and alleviating associated physiological symptoms.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If CAR T-cell therapy is administered to treat cancer, then cancer targeting and therapeutic effectiveness is improved, but cytokine release syndrome (CRS) side effects worsen

Engineering Contradiction:
Improvetherapeutic effectivenessVSAvoidCRS side effects
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent applies preliminary action by administering prostacyclin/prostaglandin analogs (such as beraprost) before CAR T-cell infusion to prevent CRS development. The prostacyclin analog is given at a predetermined dose (e.g., 10-50 μg/day) starting 1-7 days before CAR T-cell administration and continuing for 7-14 days after, which proactively mitigates the harmful cytokine release effect before it can fully develop, while preserving the anti-tumor efficacy of CAR T-cells

Inventive Principle:
Principle #10Preliminary action

2Object-affected harmful factors

If prostacyclin/prostaglandin analogs are administered to reduce CRS, then harmful side effects are reduced, but treatment complexity increases

Engineering Contradiction:
ImproveCRS side effectsVSAvoidtreatment protocol
Core Design Contradiction:
Object-affected harmful factorsVSDevice complexity

Solution Approach 1:

The patent applies parameter changes by using prostacyclin/prostaglandin analogs with specific pharmacological properties (long half-life, selective receptor binding) to reduce CRS. The treatment protocol specifies precise dosing parameters (10-50 μg/day), timing parameters (1-7 days before CAR T-cell infusion, continuing 7-14 days after), and route parameters (subcutaneous or intravenous administration), which standardize the complex interaction between the analog and CAR T-cells to achieve consistent CRS reduction

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentUS20240398947A1Car t-cell adjuvant therapies
Publication Date: 2024.12.05 CYTOAGENTS INC

AI summary

Compositions, methods, and kits that can be used to treat cancer are described herein. For example, pharmaceutical compositions containing beraprost or salts thereof can be used as an adjuvant therapy with chimeric antigen receptor T-cells (CAR T-cells) to treat cancer while reducing or eliminating undesired and potentially dangerous cytokine release syndrome (CRS) effects.