Beta Cell Biomarker Imaging for Non-Invasive Diabetes Monitoring

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Solution Overview

Problem

Current methods for imaging and quantifying pancreatic beta cell mass in diabetes are inadequate, as they rely on invasive procedures and lack specificity, making it difficult to accurately follow beta cell mass in diabetic patients and predict disease progression or response to therapies.

Innovation Solution

A biomarker specifically expressed on beta cells, such as DPP6, is used for non-invasive imaging and targeting strategies, allowing for the visualization and quantification of beta cell mass through labeled antibodies or peptides, enabling early identification of beta cell mass variations and monitoring of diabetes therapies.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If invasive procedures are used to determine beta cell mass, then measurement precision may be improved, but ease of operation deteriorates and loss of time increases

Engineering Contradiction:
Improvebeta cell mass measurement precisionVSAvoidprocedure invasiveness
Core Design Contradiction:
Measurement precisionVSEase of operation

Solution Approach 1:

The patent replaces invasive mechanical/biological procedures (pancreatectomy, autopsy, biopsy) with non-invasive molecular imaging techniques. Radioligands bind to beta-cell-specific biomarkers and are detected by imaging modalities (PET, SPECT, MRI), eliminating the need for tissue removal while maintaining measurement capability.

Inventive Principle:
Principle #28Mechanics substitution (Replace mechanical system)

Solution Approach 2:

The patent introduces radioligands as intermediary molecules that specifically bind to beta-cell biomarkers. These radioligands serve as mediators between the imaging system and beta cells, enabling indirect detection of beta cell mass without direct tissue sampling.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Ease of operation

If general imaging methods are used, then ease of operation is maintained, but measurement precision of beta cell mass deteriorates

Engineering Contradiction:
Improveimaging accessibilityVSAvoidbeta cell mass measurement precision
Core Design Contradiction:
Ease of operationVSMeasurement precision

Solution Approach 1:

The patent applies local quality by using radioligands with high specificity for beta-cell biomarkers. The radioligands concentrate specifically in beta cells rather than distributing uniformly, enabling precise localization and quantification of beta cell mass within the pancreas while maintaining ease of whole-body imaging.

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The patent uses radioligands labeled with radioactive isotopes or contrast agents that produce detectable signals (analogous to color changes). The signal intensity correlates with beta cell mass, allowing precise quantification through standard imaging modalities without requiring specialized equipment.

Inventive Principle:
Principle #32Color changes

3Device complexity

If current imaging methods are used, then device complexity is minimized, but reliability of beta cell mass determination deteriorates

Engineering Contradiction:
Improveimaging system complexityVSAvoidbeta cell mass determination reliability
Core Design Contradiction:
Device complexityVSReliability

Solution Approach 1:

The patent changes the biochemical parameter being measured by targeting specific beta-cell biomarkers (e.g., synaptotagmin, chromogranin) rather than using non-specific tracers. This biomarker-specific approach increases reliability of beta cell mass determination while using standard imaging equipment, without requiring complex new devices.

Inventive Principle:
Principle #35Parameter changes

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach enables early prediction and intervention in diabetes, allows for the follow-up of beta cell mass after islet transplantation, and provides a non-invasive method for diagnosing and monitoring diabetic disorders by detecting beta cell mass, potentially leading to better treatment strategies.

Implementation Method 1

A biomarker specifically expressed on beta cells, such as DPP6, is used for non-invasive imaging and targeting strategies, allowing for the visualization and quantification of beta cell mass through labeled antibodies or peptides

Methodology Applied
Scientific EffectAntibody-antigen binding:

Data Source

PatentEP3446126B1A new biomarker expressed in pancreatic beta cells useful in imaging or targeting beta cells
Publication Date: 2024.06.12 UNIV LIBRE DE BRUXELLES
  • EP3446126B1 patent drawingFigure 1
  • EP3446126B1 patent drawingFigure 2~3
  • EP3446126B1 patent drawingFigure 4A~4B

AI summary

The present invention is directed to the identification of a biomarker specifically located in the plasma membrane of pancreatic beta cells. Based on a set of specific features the biomarker is a unique candidate for imaging and targeting strategies to study the pancreatic beta cell mass in health and disease (T1D, T2D, pancreatic cancers, obesity, islet transplantation, beta cell regeneration).