Photoactivated Borate Bleaching for Multiplex Biological Detection

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Solution Overview

Problem

Current methods for analyzing biological samples are limited in their ability to detect multiple targets simultaneously due to fluorescence-based detection systems, requiring additional samples and struggling with the stability and efficiency of borate compounds used for signal bleaching, especially with xanthene dyes.

Innovation Solution

A novel method employing a signal cycling process with a borate compound acting as an electron transfer agent for photo-induced chemical bleaching, allowing the reuse of fluorescent dyes to detect multiple markers in a biological sample by irradiating with visible light, effectively bleaching xanthene dyes without the need for special storage or handling.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If anionic borates with cationic counter ion are used for photobleaching, then bleaching efficiency is improved, but stability to oxidation deteriorates and special storage/handling is required

Engineering Contradiction:
Improvebleaching efficiencyVSAvoidstability to oxidation
Core Design Contradiction:
ProductivityVSReliability

Solution Approach 1:

The patent changes the chemical parameters of the borate compound by introducing bulky hydrophobic groups (such as t-butyl groups) and adjusting the charge distribution. This modifies the borate's chemical stability while maintaining its photobleaching capability, allowing it to resist oxidation without requiring special storage conditions.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite structure within the borate molecule by combining electron-withdrawing groups with bulky hydrophobic groups. This composite molecular structure achieves both high bleaching efficiency and oxidation stability, resolving the contradiction between productivity and reliability.

Inventive Principle:
Principle #40Composite materials

2Productivity

If multiple targets are detected simultaneously using fluorescence-based detection, then analysis throughput is improved, but the number of detectable targets is limited by the detection system

Engineering Contradiction:
Improveanalysis throughputVSAvoidnumber of detectable targets
Core Design Contradiction:
ProductivityVSAdaptability or versatility

Solution Approach 1:

The patent employs periodic photobleaching cycles where fluorophores are sequentially activated and then bleached. This periodic action allows the same detection channel to be reused multiple times for different targets, enabling detection of many more targets than the number of simultaneously detectable fluorophores.

Inventive Principle:
Principle #19Periodic action

Solution Approach 2:

The patent temporarily discards the fluorophore signal by photobleaching it after detection, then recovers the detection channel for reuse with a different fluorophore. This cycle of discarding and recovering allows multiplexed detection beyond the limits of simultaneous fluorophore detection.

Inventive Principle:
Principle #34Discarding and recovering

3Quantity of substance

If additional biological samples are used for further analysis, then sufficient sample material is available, but sample availability is limited and sample integrity must be maintained

Engineering Contradiction:
Improvesample material availabilityVSAvoidsample reuse capability
Core Design Contradiction:
Quantity of substanceVSAdaptability or versatility

Solution Approach 1:

The patent performs preliminary detection of multiple targets in a single sample using sequential photobleaching cycles before any further analysis is needed. This preliminary multiplexed detection maximizes the information obtained from the limited sample, eliminating the need for additional samples.

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

Enables high-throughput multiplex sample analysis, allowing for the sequential detection of multiple targets with improved stability and efficiency, reducing the need for additional samples and maintaining the integrity of the biological sample.

Implementation Method 1

a photo-induced chemical bleaching (PICB) step allows the same signal generators, e.g., fluorophores, to be reused in the subsequent cycle to detect additional markers

Methodology Applied
Scientific EffectPhoto-induced chemical bleaching: Photo-oxidation

Implementation Method 2

The PICB step can include applying a borate compound of Formula I, which acts as an electron transfer agent, and initiating a photoreaction

Methodology Applied
Scientific EffectElectron transfer: Redox Reactions

Implementation Method 3

initiating a photoreaction, e.g., by irradiating the sample with visible light

Methodology Applied
Scientific EffectLight absorption: Absorption (EM radiation)

Data Source

PatentEP3256857B1Photoactivated chemical bleaching of dyes using borates
Publication Date: 2019.07.24 GENERAL ELECTRIC CO
  • EP3256857B1 patent drawingFigure 1(a)~1(e)
  • EP3256857B1 patent drawingFigure 2(a)~2(b)
  • EP3256857B1 patent drawingFigure 3(a)~3(b)

AI summary

Methods comprising the use of photoactivated chemical bleaching for detecting multiple targets in a biological sample are provided. The methods include the steps of providing a biological sample containing multiple targets, binding at least one probe to one or more target present in the sample, and observing a signal from the probe. The method further includes the steps of contacting the sample comprising the bound probe with a cationic or zwitterionic borate compound and irradiating the sample, thereby initiating a photoreaction that substantially inactivates the probe by photoactivated chemical bleaching. The method further includes the steps of binding at least one probe to one or more target present in the sample, and observing a signal from the probe. The process of binding, observing and bleaching may be iteratively repeated.