Cabergoline Antiprolactin Composition for Ruminant Dry Period Management

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Solution Overview

Problem

Shortened dry periods in ruminants lead to metabolic diseases and reproductive disorders, and previous attempts to reduce the dry period length have resulted in increased risks of these issues and decreased milk production.

Innovation Solution

Administration of a veterinary composition containing antiprolactin compounds, such as cabergoline, as dopamine receptor agonists during the dry period to prevent and reduce deleterious effects, while maintaining milk production capacity and quality.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Ease of operation

If the dry period is shortened to simplify management and reduce dietary transition time, then management complexity is reduced and lactation production period is extended, but metabolic diseases and reproductive disorders increase and milk production quality deteriorates

Engineering Contradiction:
Improvemanagement complexityVSAvoidhealth status
Core Design Contradiction:
Ease of operationVSReliability

Solution Approach 1:

The patent introduces antiprolactin compounds (dopamine receptor agonists) as intermediary substances that mediate between the shortened dry period and the ruminant's physiological needs. These compounds act as protective agents that prevent metabolic and reproductive disorders while allowing the dry period to be shortened, thus resolving the contradiction between simplified management and maintained health status

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent changes the physiological parameter of prolactin levels by administering antiprolactin compounds during the shortened dry period. This parameter change allows the animal to transition more smoothly from lactation to non-lactation state, preventing metabolic disturbances while maintaining the benefits of a shorter dry period

Inventive Principle:
Principle #35Parameter changes

2Productivity

If the dry period is shortened to extend lactation production period, then productivity is improved, but milk production capacity and quality are reduced

Engineering Contradiction:
Improvelactation production periodVSAvoidmilk production capacity
Core Design Contradiction:
ProductivityVSQuantity of substance

Solution Approach 1:

The patent applies preliminary action by administering antiprolactin compounds at the beginning of the shortened dry period. This preliminary intervention prepares the ruminant's physiology for the upcoming lactation resumption, ensuring that milk production capacity is maintained even though the dry period is shortened. The compound is given before the physiological stress of the shortened transition occurs

Inventive Principle:
Principle #10Preliminary action

3Loss of time

If the dry period is shortened to reduce dietary transition time, then loss of time is reduced, but metabolic balance is disturbed and disease risk increases

Engineering Contradiction:
Improvedry period durationVSAvoidmetabolic disease risk
Core Design Contradiction:
Loss of timeVSObject-affected harmful factors

Solution Approach 1:

The patent converts the harmful effect of the shortened dry period (metabolic imbalance) into a beneficial situation by using antiprolactin compounds to actively prevent and treat metabolic disorders. The compound transforms the potentially harmful rapid transition into a controlled physiological process, reducing disease risk while maintaining the time savings of a shorter dry period

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The use of antiprolactin compounds effectively reduces metabolic diseases and reproductive disorders, improves immune status and liver functions, and extends lactation production period without affecting milk production or quality.

Implementation Method 1

The antiprolactin compounds of the veterinary compositions of the present disclosure are chosen from dopamine receptor agonist compounds derived from ergot or from agonist compounds not derived from ergot derivatives

Methodology Applied
Scientific EffectDopamine receptor agonism:

Data Source

PatentEP2675527B1Veterinary Anti-prolactin composition for ruminants comprising cabergolin
Publication Date: 2018.10.31 CEVA SANTE ANIMALE SA
  • EP2675527B1 patent drawingFigure 1
  • EP2675527B1 patent drawingFigure 2~2B
  • EP2675527B1 patent drawingFigure 3

AI summary

The present invention relates to a veterinary anti-prolactin composition to be administered to ruminants. Said composition includes at least one anti-prolactin compound which is an agonist for dopamine receptors and which is particularly useful for preventing and/or reducing the harmful effects in ruminants linked to use for a shortened dry period. Said composition is particularly useful for preventing and/or reducing metabolic diseases and/or reproductive disorders when lactation is resumed. The use of the veterinary anti-prolactin composition according to the invention does not adversely affect the milk-producing ability and/or the milk quality of the treated ruminants.