Low-Dose Cannabinoids Prevent Cancer Cachexia

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Solution Overview

Problem

Current treatments for cancer-induced cachexia and pre-cachexia are ineffective in preventing weight loss and improving survival in cancer patients, as they fail to reverse muscle and fat wasting despite nutritional interventions and anti-inflammatory therapies.

Innovation Solution

Administering low doses of cannabinoids, such as nabilone, before and during chemotherapy, and continuing their use after chemotherapy, to inhibit the onset and progression of pre-cachexia and cachexia in cancer patients, thereby reducing weight loss and improving quality of life.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If conventional nutritional support and anti-inflammatory therapies are administered to cancer patients, then some symptomatic relief may be achieved, but weight loss and muscle wasting continue unabated

Engineering Contradiction:
Improveeffectiveness of treatmentVSAvoidweight loss
Core Design Contradiction:
ReliabilityVSLoss of substance

Solution Approach 1:

The patent changes the pharmacological parameter by introducing cannabinoids with specific receptor affinity (CB1 and CB2) to alter the metabolic and inflammatory parameters that drive cachexia, thereby preventing weight loss where conventional therapies failed

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

Cannabinoids act as intermediary substances that mediate between the harmful catabolic effects of cancer and the body's metabolic processes, blocking the progression of cachexia through receptor-mediated mechanisms

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If high doses of cannabinoids are administered to prevent cachexia, then weight loss prevention may improve, but psychoactive side effects and toxicity increase

Engineering Contradiction:
Improveprevention of weight lossVSAvoidpsychoactive side effects
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent optimizes the dosage parameter to low levels (0.1-2.5mg/day) and selects specific cannabinoid compounds with high receptor affinity, achieving effective cachexia prevention while minimizing psychoactive side effects through precise parameter control

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent applies partial action by using sub-psychoactive doses of cannabinoids that are sufficient to activate anti-cachexia mechanisms through CB1 and CB2 receptors but insufficient to produce significant psychoactive effects

Inventive Principle:
Principle #16Partial or excessive action

Data Source

PatentEP3544598B1Cannabinoids for prophylactic treatment of involuntary weight loss
Publication Date: 2021.10.06 AOP ORPHAN PHARMA AG

AI summary

The present invention provides a new use for cannabinoids in the prevention of pre-cachexia or cachexia in a patient suffering from cancer, wherein said cannabinoid is administered at low dosage and wherein administration is started prior to chemotherapy and is maintained for at least the duration of the chemotherapy.