Engineered Cas Enzyme Platform for Precise Eukaryotic Gene Editing

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Solution Overview

Problem

Current CRISPR-Cas systems lack powerful and programmable effectors for efficient genome engineering, particularly in eukaryotic cells, necessitating the development of alternative tools for modifying nucleic acids and polynucleotides.

Innovation Solution

The development of an isolated Cas enzyme with specific amino acid sequences and fusion molecules, combined with engineered guide RNAs and vector systems, to target and alter gene expression in eukaryotic cells, including mammalian cells, by binding and cleaving target DNA strands.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If CRISPR-Cas systems are used for genome engineering in eukaryotic cells, then genome editing capability is improved, but the available effector options are limited and system complexity increases

Engineering Contradiction:
Improvegenome engineering capabilityVSAvoidsystem complexity
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The patent segments the CRISPR system into distinct functional modules: guide RNA molecules for target recognition and Cas enzymes for catalytic activity. This segmentation allows independent optimization of each component and facilitates modular assembly for different applications, resolving the complexity issue while maintaining versatility.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent develops universal Cas enzyme platforms that can perform multiple functions including DNA cleavage, base editing, and epigenetic modification. By creating multi-functional effectors, the system achieves broad adaptability across different genome engineering applications without requiring separate systems for each function, thus improving versatility while managing complexity.

Inventive Principle:
Principle #6Universality (Multi-functionality)

2Productivity

If alternative programmable effectors are developed for eukaryotic cells, then efficiency of genome engineering is improved, but the available toolset remains insufficient

Engineering Contradiction:
Improvegenome engineering efficiencyVSAvoidavailable toolset
Core Design Contradiction:
ProductivityVSAdaptability or versatility

Solution Approach 1:

The patent optimizes key parameters of Cas enzymes including PAM sequence recognition, target sequence length, and catalytic activity levels. By systematically varying these parameters, the patent generates a family of effectors with different properties, thereby expanding the available toolset while maintaining high engineering efficiency across diverse applications.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates composite effector systems by fusing Cas enzymes with additional functional domains such as base editors, epigenetic modifiers, or fusion partners. These composite effectors provide enhanced functionality and expand the toolset available for eukaryotic genome engineering while maintaining efficient activity.

Inventive Principle:
Principle #40Composite materials

3Reliability

If current CRISPR-Cas systems are used, then DNA cleavage activity is achieved, but precision and control over gene expression alteration are limited

Engineering Contradiction:
ImproveDNA cleavage activityVSAvoidgene expression control precision
Core Design Contradiction:
ReliabilityVSManufacturing precision

Solution Approach 1:

The patent introduces dynamic control mechanisms through regulatable Cas enzyme systems and inducible guide RNA expression. This allows precise temporal and spatial control over when and where DNA cleavage occurs, enhancing both the reliability of cleavage activity and the precision of gene expression control by enabling on-demand activation.

Inventive Principle:
Principle #15Dynamics

Solution Approach 2:

The patent employs intermediary molecules such as base editors and epigenetic modifiers that mediate between the Cas enzyme and the target DNA. These intermediaries provide precise control over the outcome by enabling specific modifications (e.g., base conversions, methylation) without requiring double-strand breaks, thereby improving both reliability and precision simultaneously.

Inventive Principle:
Principle #24Intermediary (Mediator)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

Enables precise and efficient alteration of gene expression in eukaryotic cells, such as human cells, through the use of engineered CRISPR-Cas systems, enhancing genome engineering capabilities.

Implementation Method 1

the catalytically active domain capable of binding to a target DNA strand

Methodology Applied
Scientific EffectSequence-specific binding:

Implementation Method 2

a catalytically active domain capable of cleaving the target DNA strand

Methodology Applied
Scientific EffectCatalytic cleavage: Enzyme

Data Source

PatentEP4726035A1Cas enzyme and system and use thereof
Publication Date: 2026.04.15 EPIGENIC THERAPEUTICS PTE LTD
  • EP4726035A1 patent drawingFigure 1A
  • EP4726035A1 patent drawingFigure 1B
  • EP4726035A1 patent drawingFigure 2A~2B

AI summary

The present application relates to the field of biomedicine, and specifically relates to a novel Cas enzyme, a system thereof and the use thereof.