Casein Fusion Protein Expression via Hydrophilic Peptide Linkage

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Solution Overview

Problem

Current methods for producing milk proteins, particularly caseins, through recombinant DNA expression in heterologous hosts are not economically viable for α-S1, α-S2, and β-caseins, as established strategies like strong promoters and multiple DNA insertions are not effective for these proteins.

Innovation Solution

A recombinant fusion protein is created by combining caseins (α-S1, α-S2, or β-casein) with a caseinomacropeptide (CMP) or its fragment, which increases the hydrophilicity of the protein, improving expression yields by reducing hydrophobicity and enhancing solubility.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If strong promoters or multiple copies of recombinant DNA are used, then expression levels of κ-casein are improved, but expression levels of α-S1 casein, α-S2 casein and β-casein remain low

Engineering Contradiction:
Improveexpression levelVSAvoideffectiveness across different casein types
Core Design Contradiction:
ProductivityVSAdaptability or versatility

Solution Approach 1:

The invention uses κ-casein as an intermediary component to create fusion proteins with α-S1, α-S2, or β-casein. The κ-casein portion of the fusion protein contains sequences that are recognized by the host cell's secretion and expression machinery, thereby mediating improved expression and secretion of the otherwise poorly expressed casein variants through the fusion construct.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Ease of manufacture

If caseins are expressed alone, then the protein structure is simple, but solubility and expression yield are poor due to hydrophobicity

Engineering Contradiction:
Improveprotein simplicityVSAvoidsolubility and expression yield
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The invention creates composite fusion proteins by combining hydrophobic casein sequences with hydrophilic κ-casein sequences. This composite structure integrates the functional properties of both components: the target casein structure with the solubility-enhancing and secretion-facilitating properties of κ-casein, thereby improving expression yield and solubility while maintaining the ability to produce the desired casein variant.

Inventive Principle:
Principle #40Composite materials

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The recombinant fusion protein approach significantly increases the expression levels of caseins, making the production process more sustainable and economically viable by improving protein solubility and yield in heterologous systems.

Implementation Method 1

The peptide may increase the hydrophilicity of the recombinant fusion protein relative to the hydrophilicity of the casein alone. In other words, the peptide may decrease the hydrophobicity of the recombinant fusion protein relative to the hydrophobicity of the casein alone.

Methodology Applied
Scientific EffectHydrophilicity enhancement: Hydrophile

Data Source

PatentEP4328240A1Recombinant protein production
Publication Date: 2024.02.28 REAL DEAL MILK SL
  • EP4328240A1 patent drawingFigure 1~2b
  • EP4328240A1 patent drawingFigure 3~4
  • EP4328240A1 patent drawing

AI summary

A recombinant fusion protein is provided comprises (a) a casein selected from α-S1 casein, α-S2 casein and β-casein; and (b) a peptide comprising a caseinomacropeptide (CMP), or a fragment thereof. The recombinant fusion protein may be produced by culturing a host cell comprising a nucleic acid encoding the protein. The recombinant fusion protein finds use in the production of a recombinant casein and food compositions comprising casein.