Circular RNA Ligation Using Split RNA Elements Without Splints

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Solution Overview

Problem

Current methods for producing circular RNAs (circRNAs) with coding ability are inefficient and introduce insertions or deletions, often requiring splint oligonucleotides, leading to inaccurate ligation and polymeric by-products.

Innovation Solution

A method involving linear RNA precursors with engineered split portions forming a stable double-stranded region and a nick, ligated by RNA ligase to produce circRNAs without splint oligonucleotides, ensuring high yield and accuracy.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If T4 RNA ligase 1-mediated ligation is used to cyclize RNA, then circular RNAs can be produced, but insertions and deletions are introduced during the ligation process resulting in inaccurate ligation

Engineering Contradiction:
Improvecircular RNA productionVSAvoidligation accuracy
Core Design Contradiction:
ProductivityVSManufacturing precision

Solution Approach 1:

A splint oligonucleotide is introduced as an intermediary molecule to facilitate accurate ligation. The splint hybridizes to complementary sequences on the linear RNA ends, bringing them into proper alignment for ligation by T4 RNA ligase 1, thereby preventing insertions and deletions while enabling circular RNA formation

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The splint oligonucleotide serves as a template or copy that defines the correct spatial arrangement for ligation. By providing a predefined sequence that complements both ends of the linear RNA, it ensures that the ligation occurs at the precise intended location without introducing errors

Inventive Principle:
Principle #26Copying

2Productivity

If splint oligonucleotide is used to bring the two ends of linear RNA together for ligation, then efficient ligation can be achieved, but polymeric by-products form and the splint must be removed

Engineering Contradiction:
Improveligation efficiencyVSAvoidpolymeric by-products
Core Design Contradiction:
ProductivityVSObject-generated harmful factors

Solution Approach 1:

The harmful polymeric by-products and the splint oligonucleotide itself are extracted or removed from the final circular RNA product through purification steps, yielding clean circular RNA without contaminating sequences

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The splint oligonucleotide, after serving its purpose of facilitating ligation, is discarded or removed from the reaction mixture. The circular RNA product is recovered in a purified state, free from the splint and polymeric by-products

Inventive Principle:
Principle #34Discarding and recovering

3Ease of manufacture

If splint oligonucleotide is required for ligation, then the process can proceed, but additional sequences are introduced that may be immunogenic or reduce cargo size

Engineering Contradiction:
Improveligation feasibilityVSAvoidimmunogenicity and cargo size reduction
Core Design Contradiction:
Ease of manufactureVSObject-affected harmful factors

Solution Approach 1:

The splint oligonucleotide is designed as a temporary, disposable element that is present only during the ligation reaction. It is completely removed afterward, leaving no permanent sequence in the final circular RNA product, thus avoiding immunogenicity and cargo size issues

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The method achieves high-efficiency and accurate production of circRNAs, promoting translation of coding sequences while avoiding additional sequences that could be immunogenic or reduce cargo size.

Implementation Method 1

the first portion of the RNA element and the second portion of the RNA element associate with each other to form a double-stranded region

Methodology Applied
Scientific EffectBase pairing: Chemical Bonding

Implementation Method 2

the nick can be ligated by a RNA ligase (e.g., T4 RNA ligase 1 or T4 RNA ligase 2)

Methodology Applied
Scientific EffectEnzymatic ligation: Enzyme

Data Source

PatentEP4392560B1Constructs and methods for preparing circular RNA
Publication Date: 2026.03.11 PEKING UNIV
  • EP4392560B1 patent drawingFigure 1
  • EP4392560B1 patent drawingFigure 2A
  • EP4392560B1 patent drawingFigure 2B~2C

AI summary

Provided are linear RNA precursors and constructs for preparing circular RNAs (circRNAs) comprising from the 5' end to the 3' end: (a) a first portion of an RNA element (such as an IRES), (b) an effector RNA sequence, and (c) a second portion of the RNA element, wherein the first portion of the RNA element and the second portion of the RNA element associate with each other to form a double-stranded region of at least 4 basepairs (bp) long, wherein the 5' end of the first portion of the RNA element and the 3' end of the second portion of the RNA element form a nick in the double-stranded region, and wherein the nick can be ligated by a RNA ligase. Also provided are methods of preparing circRNAs, and circRNAs prepared thereof.