Cry1B Polypeptide Variant for Broader Lepidopteran Pest Control

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Existing genetically engineered crops provide resistance to only a narrow range of economically important insect pests, necessitating the development of new Bt toxins with improved insecticidal activity against insects from the orders Lepidoptera and Coleoptera, and biopesticides with broader activity against various insect pests.

Innovation Solution

A variant Cry1B polypeptide with an L50F amino acid substitution and a recombinant polynucleotide encoding it, operably linked to a heterologous regulatory element, is introduced into transgenic plants to enhance insecticidal activity against fall armyworm and other Lepidopteran pests.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If broad-spectrum chemical insecticides are used, then insect pest control effectiveness is improved, but environmental hazards and pollution increase

Engineering Contradiction:
Improveinsect pest control effectivenessVSAvoidenvironmental hazards
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent applies parameter changes by modifying the amino acid sequence of Cry1B polypeptide (specifically L50F substitution) to alter its insecticidal properties. This creates a variant with enhanced activity spectrum against both Lepidoptera and Coleoptera, reducing the need for broad-spectrum chemical insecticides and their associated environmental hazards.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite approach by combining the L50F amino acid substitution with existing Cry1B polypeptide structure, resulting in a hybrid variant that exhibits both the stability of the original and enhanced activity against multiple insect orders, thereby reducing reliance on hazardous chemical insecticides.

Inventive Principle:
Principle #40Composite materials

2Object-affected harmful factors

If genetically engineered crops producing Bacillus pesticidal proteins are used, then environmental friendliness is improved, but insecticidal activity spectrum is limited

Engineering Contradiction:
Improveenvironmental friendlinessVSAvoidinsecticidal activity spectrum
Core Design Contradiction:
Object-affected harmful factorsVSAdaptability or versatility

Solution Approach 1:

The patent modifies the amino acid parameters of Cry1B polypeptide by introducing the L50F substitution, which fundamentally changes the protein's activity spectrum. This single amino acid change enables the protein to effectively target both Lepidoptera and Coleoptera, expanding the versatility of environmentally friendly biopesticides.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The variant Cry1B polypeptide achieves multi-functionality by being effective against multiple insect orders (Lepidoptera and Coleoptera). This universal activity allows a single biopesticide product to replace multiple specialized products, maintaining environmental friendliness while significantly broadening the range of controlled pests.

Inventive Principle:
Principle #6Universality (Multi-functionality)

3Ease of manufacture

If standard Cry1B polypeptide is used, then production cost is reduced, but insecticidal activity against fall armyworm is insufficient

Engineering Contradiction:
Improveproduction costVSAvoidinsecticidal activity against fall armyworm
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The patent introduces a specific amino acid substitution (L50F) that optimizes the Cry1B polypeptide's activity against fall armyworm. This targeted modification enhances binding affinity or toxicity mechanism specifically for fall armyworm while maintaining relatively simple production requirements through recombinant DNA technology.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3207050B1Insecticidal polypeptides having improved activity spectrum and uses thereof
Publication Date: 2026.04.22 PIONEER HI BREED INTERNATIONAL INC
  • EP3207050B1 patent drawingFigure 1a
  • EP3207050B1 patent drawingFigure 1b
  • EP3207050B1 patent drawingFigure 1c

AI summary

The disclosure provides nucleic acids, and variants and fragments thereof, derived from strains of Bacillus thuringiensis encoding variant polypeptides having increased pesticidal activity against insect pests, including Lepidoptera and Coleopteran. Particular embodiments of the disclosure provide isolated nucleic acids encoding pesticidal proteins, pesticidal compositions, DNA constructs, and transformed microorganisms and plants comprising a nucleic acid of the embodiments. These compositions find use in methods for controlling pests, especially plant pests.