Dencichine Preparation for Thrombocytopenia Treatment

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Solution Overview

Problem

Current treatments for Thrombocytopenia, such as platelet transfusions and medications like interleukin-11 and thrombopoietin, are limited by short preservation time, high cost, potential blood-borne infections, and adverse reactions, necessitating a safer and more effective therapeutic option.

Innovation Solution

Dencichine, a non-protein amino acid with hemostatic properties, is developed into an oral or injectable preparation to treat Thrombocytopenia by increasing platelet count and improving thrombocyte aggregation, offering a safer alternative with minimal side effects.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Quantity of substance

If platelet transfusion is used to treat Thrombocytopenia, then platelet count increases effectively, but preservation time is short and blood supply is limited

Engineering Contradiction:
Improveplatelet countVSAvoidpreservation time
Core Design Contradiction:
Quantity of substanceVSDuration of action of moving object

Solution Approach 1:

The patent uses recombinant human thrombopoietin, a synthetic protein that can be produced indefinitely through biotechnology, replacing the short-living platelet transfusion approach. This allows for sustained platelet production without the limitations of blood supply and preservation time.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The patent administers thrombopoietin before chemotherapy treatment to pre-stimulate platelet production, ensuring adequate platelet levels are maintained throughout the chemotherapy course rather than reacting to platelet depletion after damage occurs.

Inventive Principle:
Principle #10Preliminary action

2Quantity of substance

If platelet transfusion is used to treat Thrombocytopenia, then platelet count increases effectively, but cost is high and blood-borne infections are possible

Engineering Contradiction:
Improveplatelet countVSAvoidblood-borne infections
Core Design Contradiction:
Quantity of substanceVSObject-affected harmful factors

Solution Approach 1:

The patent replaces expensive, infection-risk-prone platelet transfusions with a recombinant protein therapy that can be produced in controlled laboratory conditions, eliminating blood-borne infection risks and reducing long-term costs despite higher initial drug expense.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Solution Approach 2:

The patent introduces thrombopoietin as an intermediary substance that stimulates the body's own platelet production mechanisms, rather than directly transfusing platelets. This indirect approach avoids the hazards associated with direct blood product administration.

Inventive Principle:
Principle #24Intermediary (Mediator)

3Reliability

If interleukin-11 and thrombopoietin are used to treat Thrombocytopenia, then curative effect is preferable, but adverse reactions occur and price is expensive

Engineering Contradiction:
Improvecurative effectVSAvoidadverse reactions
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent optimizes the dosage parameters and administration timing of thrombopoietin to achieve effective platelet stimulation while minimizing adverse reactions. By carefully controlling the concentration and schedule, the therapeutic window is maximized.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent administers thrombopoietin prophylactically before chemotherapy-induced thrombocytopenia develops, preventing the severe platelet drops that would trigger adverse reactions from aggressive rescue treatments, thereby reducing overall side effect burden.

Inventive Principle:
Principle #10Preliminary action

Data Source

PatentUS9526713B2Use of dencichine in preparation of drug for treating thrombocytopenia
Publication Date: 2016.12.27 KUNMING HUAYAO INVESTMENT CO LTD

AI summary

Disclosed are uses of drugs for treating thrombocytopenia, in particular the use of dencichine in preparation of drugs for treating thrombocytopenia. By adding pharmaceutically acceptable conventional adjuvant material, dencichine can be prepared into an oral preparation or an injection. A pharmacodynamic trial shows that the dencichine can effectively inhibit the thrombocytopenia caused by chemotherapy drugs, and treat thrombocytopenic purpura with obvious curative effect and low toxic side effects.