Enterococcus sp. I-4969 for Asthma Th1/Th2 Cytokine Modulation

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current treatments for respiratory diseases, particularly asthma, are inadequate in effectively preventing and managing symptoms, and there is a need for compositions that can easily and effectively treat and prevent respiratory tract infections.

Innovation Solution

A specific strain of Enterococcus sp. (deposited as I-4969) is used, which limits inflammation and weight loss in animal models of chronic allergic asthma by increasing Th1 cytokine expression while reducing Th2 cytokine expression, and can be administered in live or inactivated form, either alone or with pharmaceutically acceptable excipients.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If conventional treatments are used for respiratory diseases, then symptoms can be managed, but they are inadequate in effectively preventing and managing asthma symptoms

Engineering Contradiction:
Improveeffectiveness of treatmentVSAvoidavailability of effective compositions
Core Design Contradiction:
ReliabilityVSEase of manufacture

Solution Approach 1:

The patent changes the fundamental parameter of treatment approach by introducing live bacterial strains (Enterococcus faecalis and other Lactobacillaceae family members) as therapeutic agents. This probiotic approach modifies the immune system's response to allergens, transforming the body's reaction from allergic to tolerant, thereby effectively preventing asthma symptoms rather than merely managing them.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The bacterial strains act as intermediaries between the immune system and allergens. These probiotics modulate immune responses by promoting regulatory T cell development and anti-inflammatory cytokine production, serving as a bridge that redirects the immune system's reaction to allergens from pathological to protective.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If bacterial strains are used to treat respiratory diseases, then prevention and treatment efficacy is improved, but the complexity of administering live bacteria increases

Engineering Contradiction:
Improveprevention and treatment efficacyVSAvoidadministration complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent employs probiotic bacteria that serve multiple functions: they colonize the respiratory tract, modulate immune responses, prevent allergic sensitization, and treat existing asthma symptoms. This multi-functionality simplifies the overall treatment strategy by combining prevention and treatment in a single therapeutic agent.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Solution Approach 2:

The probiotic bacteria are self-replicating and self-sustaining once administered. They colonize the respiratory tract and maintain their therapeutic effect through continuous production of immunomodulatory substances, eliminating the need for complex dosing schedules or external support systems.

Inventive Principle:
Principle #25Self-service

3Measurement precision

If metagenome studies are used to identify lung microbiota, then bacterial diversity can be detected, but the bacterial load is too low for usual culturing technologies

Engineering Contradiction:
Improvedetection of bacterial strainsVSAvoiddetectability by culturing
Core Design Contradiction:
Measurement precisionVSEase of manufacture

Solution Approach 1:

The patent changes the detection parameter from relying on high bacterial load (suitable for culturing) to utilizing metagenomic sequencing that can detect low-abundance bacteria. This parameter change enables the identification and selection of rare probiotic strains from the lung microbiota that would be invisible to traditional culturing methods.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP3408373B1Bacterial strain as agents for preventing and/or treating respiratory disorders
Publication Date: 2020.01.01 INST NAT DE RECH POUR LAGRICULTURE
  • EP3408373B1 patent drawingFigure 1A~1B
  • EP3408373B1 patent drawingFigure 1C
  • EP3408373B1 patent drawingFigure 1D~1E

AI summary

The invention relates to a novel bacterial strain deposited with the CNCM under number 1-4969. This strain has properties that are useful in the treatment of respiratory disorders. The invention also relates to compositions and uses of said strain.