Enzymatic Detection of 5hmC and 5mC Modifications

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Solution Overview

Problem

Current methods for analyzing DNA methylation patterns, such as sodium bisulfite sequencing, struggle to distinguish between 5-methylcytosine (5mC) and 5-hydroxymethylcytosine (5hmC) and require high DNA amounts and sequencing depth, while long-read amplicon sequencing is limited to specific genomic regions, hindering the study of the whole methylome and hydroxymethylome.

Innovation Solution

A method involving enzymatic conversion and whole genome sequencing library preparation, where DNA is fragmented, protected, denatured, and deaminated to convert cytosines into uracils, allowing for the detection and discrimination of 5mC and 5hmC without the need for expensive oligos, enabling analysis of the whole genome.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If sodium bisulfite sequencing is used to analyze DNA methylation, then methylation patterns can be detected, but the method cannot distinguish between 5mC and 5hmC and requires high DNA amounts and sequencing depth

Engineering Contradiction:
Improvedetection of methylation patternsVSAvoidDNA amount required
Core Design Contradiction:
Measurement precisionVSQuantity of substance

Solution Approach 1:

The patent segments the detection process into separate enzymatic reactions: one reaction specifically converts 5mC to uracil while leaving 5hmC unchanged, and another reaction converts both 5mC and 5hmC to uracil. By comparing the results of these segmented reactions, the method can distinguish between the two modifications without requiring high DNA amounts, as each reaction processes the sample independently and efficiently.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent introduces enzymatic intermediaries (specifically uracil DNA glycosylase and APOBEC1) that mediate the conversion of methylated cytosines to uracils. These enzymes act as selective intermediaries that can differentiate between 5mC and 5hmC based on their chemical properties, enabling precise detection without direct sequencing of the modified bases.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Measurement precision

If long-read amplicon sequencing is used to detect 5mC and 5hmC, then single-base resolution can be achieved, but the method is restricted to analysis of a few genomic regions

Engineering Contradiction:
Improvesingle-base resolutionVSAvoidgenomic region coverage
Core Design Contradiction:
Measurement precisionVSAdaptability or versatility

Solution Approach 1:

The patent creates a universal enzymatic conversion system that can process the entire genome. The enzymes (uracil DNA glycosylase and APOBEC1) act throughout the whole genome simultaneously, converting all 5mC and 5hmC sites to uracils regardless of their location. This universal approach allows subsequent sequencing to cover the entire methylome and hydroxymethylome at single-base resolution, eliminating the need for region-specific amplicon sequencing.

Inventive Principle:
Principle #6Universality (Multi-functionality)

3Ease of manufacture

If conventional library preparation methods are used, then sequencing libraries can be prepared, but expensive DNA oligos are required

Engineering Contradiction:
Improvelibrary preparationVSAvoidcost of DNA oligos
Core Design Contradiction:
Ease of manufactureVSQuantity of substance

Solution Approach 1:

The patent employs inexpensive, readily available enzymes (uracil DNA glycosylase and APOBEC1) as disposable reagents that can be easily replaced. These enzymes perform the critical function of converting methylated cytosines to uracils without requiring expensive synthetic oligos. The enzymatic reactions can be performed with standard laboratory reagents, significantly reducing the cost of library preparation while maintaining high detection accuracy.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This method effectively detects and discriminates 5mC and 5hmC across the whole genome, reducing costs and improving analysis efficiency, particularly suitable for low-input samples like circulating cell-free DNA and single-cell analysis.

Implementation Method 1

performing enzymatic deamination of the ssNA product obtained in step d1) to convert cytosines (C) and methylated cytosines (5mC) into uracils (U)

Methodology Applied
Scientific EffectEnzymatic deamination: Enzyme

Implementation Method 2

denaturing the product of step b) to obtain a modified single stranded nucleic acid sample (ssNA)

Methodology Applied
Scientific EffectHeat denaturation: Heating

Data Source

PatentEP4296372A1Method to detect and discriminate cytosine modifications
Publication Date: 2023.12.27 UNIV POMPEU FABRA (UPF)
  • EP4296372A1 patent drawingFigure 1
  • EP4296372A1 patent drawingFigure 2A~2B
  • EP4296372A1 patent drawingFigure 3A~3C

AI summary

The present invention discloses a method to detect 5-hydroxymethylcytosine (5hmC) and discriminate between 5-methylcytosine (5mC) and 5-hydroxymethylcytosine (5hmC) from a nucleic acid that comprises enzymatic treatment and construction of nucleic acid library and a kit to perform said method.