Galactose-Fucose Monosaccharide Composition for Re-Epithelialization

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Solution Overview

Problem

Existing wound and lesion treatments, including polysaccharides and growth factors, lack effective strategies to accelerate healing, minimize scarring, and enhance re-epithelialization, with monosaccharides like galactose and fucose being overlooked for their therapeutic potential due to assumptions about structural stability and enzymatic breakdown requirements.

Innovation Solution

A composition comprising galactose and fucose in monosaccharide form is used as a promotor of tissue re-epithelialization, administered topically or in various formulations to enhance cellular proliferation and healing, leveraging their natural occurrence and bioavailability.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If polysaccharides are used for wound healing, then structural stability is maintained, but re-epithelialization promotion is insufficient

Engineering Contradiction:
Improvestructural stabilityVSAvoidre-epithelialization promotion
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The patent segments the polysaccharide structure into individual monosaccharide units (galactose and fucose), allowing each unit to independently promote re-epithelialization while maintaining overall therapeutic effectiveness. This segmentation enables better absorption and cellular utilization compared to intact polysaccharides.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent changes the molecular size parameter from large polysaccharide molecules to small monosaccharide units, improving bioavailability and cellular uptake. This parameter change allows the substances to penetrate cell membranes more effectively and stimulate re-epithelialization without compromising safety.

Inventive Principle:
Principle #35Parameter changes

2Productivity

If polysaccharides are broken down to monosaccharides, then re-epithelialization is enhanced, but structural stability is compromised

Engineering Contradiction:
Improvere-epithelialization promotionVSAvoidstructural stability
Core Design Contradiction:
ProductivityVSStability of the object's composition

Solution Approach 1:

Instead of breaking down polysaccharides to monosaccharides and risking stability loss, the patent inverts the approach by directly using monosaccharides as the active therapeutic agents. This inversion eliminates the need for enzymatic breakdown in the wound site while maintaining structural integrity through the use of stable, naturally occurring monosaccharide molecules.

Inventive Principle:
Principle #13The other way round (Inversion)

3Productivity

If growth factors and cytokines are used, then healing is accelerated, but complexity and cost increase

Engineering Contradiction:
Improvehealing accelerationVSAvoidtreatment complexity
Core Design Contradiction:
ProductivityVSDevice complexity

Solution Approach 1:

The patent uses simple, naturally occurring monosaccharides (galactose and fucose) that are inexpensive to produce and administer, replacing complex and costly growth factors and cytokines. These monosaccharides provide effective healing promotion without the complexity of protein-based therapies, making them more suitable for routine wound care applications.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

4Reliability

If polysaccharides are used, then treatment is safe, but healing acceleration is limited

Engineering Contradiction:
ImprovesafetyVSAvoidhealing acceleration
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The patent changes the molecular parameter from large polysaccharide molecules to small monosaccharide units, improving cellular uptake and healing acceleration while maintaining safety. The monosaccharides are naturally occurring substances with well-established safety profiles, eliminating the need for extensive safety testing while achieving faster healing results.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentEP4659751A1Galactose and fucose monosaccharides for re-epithelialization and treating lesions
Publication Date: 2025.12.10 PATHOBLOCK THERAPEUTICS GMBH & CO KG
  • EP4659751A1 patent drawingFigure 1
  • EP4659751A1 patent drawingFigure 2
  • EP4659751A1 patent drawingFigure 3

AI summary

Disclosed is a composition (204) comprising galactose and fucose in monosaccharide form for use as a promotor of tissue re-epithelialization.