Glufosinate and Pyroxasulfone Herbicidal Composition for Broadleaf Weed Control

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Solution Overview

Problem

Current herbicidal compositions for preplant burndown, particularly those using glyphosate or glufosinate, often yield unsatisfactory weed control, especially against difficult-to-control broadleaf species and rhizomatous grasses, requiring high dosages and being weather-dependent, with limited persistence and potential toxicity to mammals.

Innovation Solution

A herbicidal composition combining glyphosate or glufosinate with pyroxasulfone and additional herbicides from specific inhibitor groups (ALS, PPO, auxins, HPPD, PSII, etc.) to enhance weed control efficacy, persistence, and safety, allowing for flexible application and reduced toxicity.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Ease of manufacture

If glyphosate or glufosinate is applied solo for burndown, then application simplicity is maintained, but weed control effectiveness deteriorates (unsatisfactory control of broadleaf species and rhizomatous grasses)

Engineering Contradiction:
Improveapplication simplicityVSAvoidweed control effectiveness
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The patent combines glyphosate or glufosinate with pyroxasulfone and additional herbicides from specific inhibitor groups (ALS, PPO, auxins, HPPD, PSII) to create a multi-component herbicidal composition. This merging of multiple herbicides with different modes of action achieves synergistic effects that improve weed control effectiveness against difficult-to-control species while maintaining practical application feasibility

Inventive Principle:
Principle #5Merging (Combining)

2Reliability

If high dosage rates of glyphosate or glufosinate are applied to improve weed control, then weed control effectiveness improves, but toxicity to mammals increases

Engineering Contradiction:
Improveweed control effectivenessVSAvoidtoxicity to mammals
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent changes the chemical composition parameters by introducing pyroxasulfone and other herbicides with different modes of action. This parameter change allows achieving effective weed control at lower overall dosage rates, thereby reducing mammalian toxicity while maintaining or improving weed control effectiveness through synergistic interactions among the herbicide components

Inventive Principle:
Principle #35Parameter changes

3Duration of action of stationary object

If conventional herbicide combinations are applied to improve weed control persistence, then persistence is extended, but reliability under varying weather conditions deteriorates (weather-dependent effectiveness)

Engineering Contradiction:
Improveherbicidal activity persistenceVSAvoidconsistency under weather conditions
Core Design Contradiction:
Duration of action of stationary objectVSReliability

Solution Approach 1:

The patent creates a composite herbicidal formulation containing glyphosate or glufosinate combined with pyroxasulfone and additional herbicides from multiple inhibitor groups. This composite material approach provides consistent herbicidal activity persistence across varying weather conditions by leveraging the complementary properties and different modes of action of the constituent herbicides

Inventive Principle:
Principle #40Composite materials

4Reliability

If multiple herbicides are combined to improve weed control spectrum, then weed control effectiveness improves, but composition complexity increases

Engineering Contradiction:
Improveweed control spectrumVSAvoidcomposition complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent designs a multi-functional herbicidal composition where pyroxasulfone and additional herbicides from specific inhibitor groups serve multiple purposes: they provide pre-emergence and post-emergence activity, target different weed species (broadleaf and grass), and offer complementary modes of action. This multi-functionality approach broadens the weed control spectrum while managing composition complexity through strategic selection of synergistic partners

Inventive Principle:
Principle #6Universality (Multi-functionality)

Data Source

PatentUS12059004B2Herbicidal composition comprising glufosinate or salt thereof and pyroxasulfone
Publication Date: 2024.08.13 BASF SE
  • US12059004B2 patent drawing
  • US12059004B2 patent drawing
  • US12059004B2 patent drawing

AI summary

The present invention relates to a herbicidal composition which comprises:a) at least one herbicide A selected from glyphosate, glufosinate and their salts, andb) a herbicide B which is 3-[5-(difluoromethoxy)-1-methyl-3-(trifluoromethyl)pyrazol-4-ylmethylsulfonyl]-4,5-dihydro-5,5-dimethyl-1,2-oxazole [common name: pyroxasulfone].The present invention relates in particular to a herbicidal composition comprising:a) at least one herbicide A selected from glyphosate, glufosinate and their salts,b) a herbicide B which is 3-[5-(difluoromethoxy)-1-methyl-3-(trifluoromethyl)pyrazol-4-ylmethylsulfonyl]-4,5-dihydro-5,5-dimethyl-1,2-oxazole [common name: pyroxasulfone], andc) at least one further herbicide C, which is selected from the herbicide groups C.1 to C.8:C.1 herbicides of the group of acetolactate synthase inhibitors (ALS inhibitors),C.2 herbicides of the group of protoporphyrinogen oxidase inhibitors (PPO inhibitors),C.3 herbicides of the group of auxines,C.4 herbicides of the group of 4-hydroxyphenyl-pyruvate-dioxygenase inhibitors (HPPD inhibitors),C.5 herbicides of the group of phytoene desaturase inhibitors (PDS inhibitors),C.6 herbicides of the group of photosystem II inhibitors (PSII inhibitors),C.7 herbicides of the group of microtubulin inhibitors, andC.8 herbicides of the group of inhibitors of the synthesis of very long chain fatty acids (VLCFA inhibitors).