Goserelin Implant Regimen Switching for Breast Cancer Adherence

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Solution Overview

Problem

Existing goserelin implant dosing regimens for breast cancer treatment face challenges in patient compliance and require frequent administration, leading to potential nonadherence and increased healthcare visits.

Innovation Solution

A dosing regimen that involves concomitant administration of a 3.6 mg goserelin acetate implant with chemotherapy cycles, followed by a switch to a 10.8 mg implant every 84 to 108 days for improved compliance and reduced frequency of administration, addressing nonadherence and enhancing treatment duration.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If a 3.6 mg goserelin implant is administered monthly, then ovarian suppression is maintained, but patient compliance deteriorates due to frequent administration requirements

Engineering Contradiction:
Improveovarian suppression efficacyVSAvoidpatient compliance
Core Design Contradiction:
ReliabilityVSEase of operation

Solution Approach 1:

The treatment regimen is segmented into two phases: an initial phase with 3.6 mg monthly implants to establish ovarian suppression, followed by a maintenance phase with 10.8 mg quarterly implants. This segmentation allows the treatment to adapt to patient compliance patterns while maintaining therapeutic efficacy.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The dosing regimen dynamically transitions from frequent monthly administrations to less frequent quarterly administrations after the initial phase. This dynamic adjustment maintains suppression efficacy while reducing the burden on patients, thereby improving compliance.

Inventive Principle:
Principle #15Dynamics

2Reliability

If a 3.6 mg goserelin implant is administered monthly, then hormone receptor positive breast cancer is treated, but treatment duration deteriorates due to patient nonadherence

Engineering Contradiction:
Improvecancer treatment efficacyVSAvoidtreatment duration
Core Design Contradiction:
ReliabilityVSDuration of action of stationary object

Solution Approach 1:

The initial phase of monthly 3.6 mg administrations serves as a preliminary action to establish reliable ovarian suppression and treatment response before transitioning to the maintenance phase. This preliminary establishment of efficacy ensures that when the dosing interval is extended, the therapeutic benefit is already secured.

Inventive Principle:
Principle #10Preliminary action

3Ease of operation

If a 10.8 mg goserelin implant is administered quarterly, then patient compliance improves, but the regimen is not approved for breast cancer treatment in the US

Engineering Contradiction:
Improvepatient complianceVSAvoidregimen approval status
Core Design Contradiction:
Ease of operationVSReliability

Solution Approach 1:

The regimen segments the use of the 10.8 mg implant into a maintenance phase following initial 3.6 mg administrations. This segmentation allows the higher-dose, longer-interval implant to be used in a controlled manner that addresses compliance issues while managing regulatory considerations.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The regimen changes the dosing parameters from 3.6 mg monthly to 10.8 mg quarterly after the initial phase. This parameter change optimizes compliance by reducing administration frequency while maintaining therapeutic effect through the cumulative dosing strategy.

Inventive Principle:
Principle #35Parameter changes

4Reliability

If frequent monthly administrations are required, then ovarian suppression is maintained, but healthcare utilization increases

Engineering Contradiction:
Improvesuppression maintenanceVSAvoidhealthcare utilization efficiency
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The regimen dynamically adjusts the administration frequency from monthly to quarterly after the initial phase. This dynamic change reduces the number of healthcare visits required for implantation and monitoring, thereby improving healthcare utilization efficiency while maintaining suppression through the optimized dosing interval.

Inventive Principle:
Principle #15Dynamics

Data Source

PatentUS20250367261A1Goserelin implant dosing regimens for improved patient compliance
Publication Date: 2025.12.04 TERSERA THERAPEUTICS LLC

AI summary

Described herein are methods of treating hormone receptor positive breast cancer in a patient which include concomitantly administering an initial neoadjuvant or adjuvant IV chemotherapy cycle and an initial dose of a 3.6 mg goserelin acetate implant to the patient, or concomitantly administering an initial dose of a 3.6 mg goserelin acetate implant to the patient with a first of a plurality of long-term IV chemotherapy cycles. After one or more doses of the 3.6 mg goserelin acetate implant, the 3.6 mg goserelin acetate implant is discontinued, and the patient is then administered a 10.8 mg goserelin implant once every 84 to 108 days. Also included are methods of improving patient compliance, increasing duration of treatment, and/or reducing the need for oophorectomy in a patient with hormone receptor positive breast cancer by administering a 3.6 mg goserelin acetate implant to the patient, and upon the patient becoming nonadherent, the 3.6 mg goserelin acetate implant is discontinued, and the patient is then administered a 10.8 mg goserelin implant once every 84 to 108 days.