Poly-allylamine Coatings with Guanidine Groups for Anti-biofilm

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Solution Overview

Problem

Current prophylactic approaches for preventing biofilm formation on teeth surfaces, such as positively charged polymeric coatings, often lead to increased bacterial adhesion due to electrostatic interactions, and existing antimicrobial coatings are not effective in the long term.

Innovation Solution

Development of an antimicrobial or antibacterial composition featuring a cationic polymer with a poly-allylamine backbone functionalized with guanidine and optionally biguanide groups, which is deposited on surfaces to inhibit microbial adhesion, using a method that includes physical adsorption and potential cross-linking with anionic polymers.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If positively charged polymeric coatings are deposited on tooth surfaces to prevent biofilm formation, then short-term prophylactic efficacy is improved, but bacterial adhesion increases due to electrostatic interactions with negatively charged bacterial cell walls

Engineering Contradiction:
Improveprophylactic efficacyVSAvoidbacterial adhesion
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent modifies the chemical structure of polymeric coatings by incorporating guanidine and biguanide functional groups into the polymer backbone. These functional groups provide broad-spectrum antimicrobial activity through mechanism independent of electrostatic charge, thereby maintaining prophylactic efficacy while eliminating the harmful effect of increased bacterial adhesion associated with positively charged coatings

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The invention uses composite polymeric structures combining multiple functional groups (guanidine, biguanide, and other antimicrobial moieties) within a single coating system. This composite approach enables simultaneous achievement of long-term durability and broad-spectrum antimicrobial activity without relying on electrostatic charge, thus resolving the contradiction between short-term efficacy and bacterial adhesion

Inventive Principle:
Principle #40Composite materials

2Reliability

If traditional prophylactic approaches are used to reduce biofilm formation, then initial protection is achieved, but the effect is only temporary and not durable

Engineering Contradiction:
Improvebiofilm preventionVSAvoidcoating durability
Core Design Contradiction:
ReliabilityVSDuration of action of stationary object

Solution Approach 1:

The patent employs polymers with enhanced chemical stability and resistance to enzymatic degradation by incorporating stable backbone structures and chemically robust functional groups. This modification extends the duration of action of the coating from short-term to long-term while maintaining effective biofilm prevention

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The antimicrobial functional groups in the polymer coating provide continuous broad-spectrum antimicrobial activity over extended periods. The coating maintains its protective function continuously rather than requiring reapplication, achieving both reliable biofilm prevention and long-term durability

Inventive Principle:
Principle #20Continuity of useful action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The cationic polymer composition effectively reduces bacterial adherence on teeth surfaces, providing a durable and long-lasting solution to biofilm prevention, outperforming traditional anionic polymers and hybrid coatings in anti-attachment capabilities.

Implementation Method 1

increased bacterial adhesion due to the negatively charged bacterial cell wall

Methodology Applied
Scientific EffectElectrostatic interactions: Electrostatics

Implementation Method 2

contacting the substrate with a first polymer to physically adsorb the first polymer to surfaces of the substrate

Methodology Applied
Scientific EffectPhysical adsorption: Adsorption

Data Source

PatentEP3512607B1Antimicrobial compositions for oral care or cleansing, and methods for Anti-attachment polymers and coatings
Publication Date: 2024.02.14 COLGATE PALMOLIVE CO
  • EP3512607B1 patent drawingFigure 1A~1B
  • EP3512607B1 patent drawingFigure 1C~1D
  • EP3512607B1 patent drawingFigure 2A~2B

AI summary

Antimicrobial compositions and methods for depositing or coating the antimicrobial or antibacterial compositions on a substrate to prevent microbial adhesion are provided. The antimicrobial composition may include a cationic polymer having a poly-allylamine backbone. A portion of the poly-allylamine backbone may be functionalized with at least one of a guanidine functional group and a biguanide functional group.