Guide RNA 5' End Tuning for Precise Transcription Control

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Solution Overview

Problem

There is a need for further technological development in controlling RNA transcription and applying RNA-guided nucleases, with a focus on designing expression vectors and kits for enhanced control over transcription and genome editing.

Innovation Solution

The method involves adding three or more nucleotide residues to the 5' end of guide RNA and adjusting the spacer sequence to control transcription and editing, utilizing RNA-guided nucleases like Cas proteins from Type V CRISPR/Cas systems, and incorporating fusion proteins with transcription regulation domains for targeted gene control.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Measurement precision

If nucleotide residues are added to the 5' end of guide RNA to control transcription, then transcription control precision is improved, but guide RNA structure complexity increases

Engineering Contradiction:
Improvetranscription control precisionVSAvoidguide RNA structure complexity
Core Design Contradiction:
Measurement precisionVSDevice complexity

Solution Approach 1:

The patent applies parameter changes by modifying the 5' end of guide RNA with specific nucleotide residues (such as uracil, cytosine, guanine, or adenine) to control transcription. By changing the nucleotide composition and sequence at the 5' end, the invention achieves precise control over transcription without fundamentally altering the overall guide RNA structure, thus resolving the contradiction between control precision and structural complexity.

Inventive Principle:
Principle #35Parameter changes

2Productivity

If spacer sequence is adjusted to enhance editing efficiency, then genome editing efficiency is improved, but off-target effects increase

Engineering Contradiction:
Improvegenome editing efficiencyVSAvoidoff-target effects
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent applies local quality by carefully designing and adjusting specific regions of the spacer sequence while maintaining the overall functionality of the guide RNA. By optimizing local nucleotide compositions and sequences in the spacer region, the invention enhances editing efficiency at the target site while minimizing off-target effects through localized sequence-specific binding, thus resolving the contradiction between editing efficiency and off-target effects.

Inventive Principle:
Principle #3Local quality

3Adaptability or versatility

If RNA-guided nucleases are used for transcription control, then transcription regulation capability is improved, but system complexity increases

Engineering Contradiction:
Improvetranscription regulation capabilityVSAvoidsystem complexity
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The patent applies universality by utilizing RNA-guided nucleases that can perform multiple functions including transcription control, genome editing, and base editing. By designing a versatile system where the same core components (guide RNA with modified 5' end and RNA-guided nuclease) can be applied to different transcription regulation scenarios, the invention enhances transcription regulation capability while avoiding the need for entirely separate systems for each application, thus reducing overall system complexity.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This approach enables precise control over RNA transcription and genome editing, enhancing the efficiency and specificity of RNA-guided nuclease applications, including base editing and transcription regulation.

Implementation Method 1

The Cas9-crRNA-tracrRNA complex binds to foreign invasive DNA complementary to the crRNA

Methodology Applied
Scientific EffectBase pairing:

Implementation Method 2

a step of transcribing RNA from an expression vector for the RNA

Methodology Applied
Scientific EffectTranscription:

Implementation Method 3

the RNA is RNA to which one or more nucleotide residues are added at the 5' end

Methodology Applied
Scientific EffectChemical modification:

Data Source

PatentEP4678745A1Guide RNA and use method thereof
Publication Date: 2026.01.14 KYUSHU UNIV
  • EP4678745A1 patent drawingFigure 1~2
  • EP4678745A1 patent drawingFigure 3
  • EP4678745A1 patent drawingFigure 4

AI summary

Provided is a method for controlling transcription of RNA, including: a step of transcribing RNA from an expression vector for the RNA, in which the RNA is RNA to which one or more nucleotide residues are added at the 5' end, and the like. In addition, provided is a method for designing an expression vector for RNA, including: designing an expression vector for RNA in which transcription efficiency of the RNA is controlled by adjusting one or more selected from the group consisting of the number of nucleotide residues to be added to the 5' end of an RNA coding sequence and the type of the nucleotide residues, and the like.