Herbicidal Composition Synergy 3-Phenyluracils

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Solution Overview

Problem

Current herbicidal compositions comprising 3-phenyluracils and 3-sulfonylisoxazolines often fail to effectively control harmful plants without damaging desirable crop plants, such as cotton, oilseed rape, and certain graminaceous plants, necessitating reduced application rates that compromise weed control efficacy.

Innovation Solution

Formulating herbicidal compositions that combine 3-phenyluracils of specific structural formulas with 3-sulfonylisoxazolines and optional safeners, which are applied in a way that enhances herbicidal activity through synergism, allowing for lower application rates while improving compatibility with useful plants.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Object-affected harmful factors

If 3-phenyluracils and 3-sulfonylisoxazolines are applied at standard rates to control harmful plants, then weed control efficacy is improved, but damage to useful crop plants increases

Engineering Contradiction:
Improveweed control efficacyVSAvoiddamage to useful crop plants
Core Design Contradiction:
Object-affected harmful factorsVSObject-generated harmful factors

Solution Approach 1:

The patent combines 3-phenyluracils and 3-sulfonylisoxazolines into a single herbicidal composition, leveraging synergistic effects to enhance weed control efficacy while reducing the need for high application rates that would damage crop plants. This merging of two active compounds allows for more precise and effective weed management at lower concentrations.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The patent modifies the chemical structure and concentration parameters of the herbicidal composition by incorporating specific substituents (R1-R9 variables) and adjusting the ratio of 3-phenyluracil to 3-sulfonylisoxazoline, thereby optimizing the balance between weed control effectiveness and crop plant safety.

Inventive Principle:
Principle #35Parameter changes

2Object-generated harmful factors

If application rates are reduced to protect useful plants, then crop plant compatibility is improved, but weed control activity is compromised

Engineering Contradiction:
Improvecompatibility with useful plantsVSAvoidweed control activity
Core Design Contradiction:
Object-generated harmful factorsVSObject-affected harmful factors

Solution Approach 1:

By merging 3-phenyluracils and 3-sulfonylisoxazolines into a combined composition, the patent achieves synergistic enhancement of weed control activity, allowing effective weed management at lower application rates that do not compromise crop plant compatibility. The combination creates a more efficient herbicidal system than either compound alone.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The patent creates a composite herbicidal composition containing both 3-phenyluracil and 3-sulfonylisoxazoline compounds, where the synergistic interaction between the two active ingredients produces enhanced weed control efficacy at reduced concentrations, thereby protecting crop plants from damage.

Inventive Principle:
Principle #40Composite materials

3Device complexity

If single herbicide compounds are used to simplify formulation, then device complexity is reduced, but herbicidal activity and selectivity are insufficient

Engineering Contradiction:
Improveformulation simplicityVSAvoidherbicidal activity and selectivity
Core Design Contradiction:
Device complexityVSObject-affected harmful factors

Solution Approach 1:

The patent merges two herbicidal compounds (3-phenyluracil and 3-sulfonylisoxazoline) into a single formulated composition, creating a synergistic system that enhances both herbicidal activity and selectivity. This combined approach provides superior weed control and crop safety compared to using either compound alone, while maintaining practical formulation simplicity.

Inventive Principle:
Principle #5Merging (Combining)

Data Source

PatentUS8889593B2Herbicidal compositions based on 3-phenyluracils and 3-sulfonylisoxazolines
Publication Date: 2014.11.18 BASF SE
  • US8889593B2 patent drawing
  • US8889593B2 patent drawing
  • US8889593B2 patent drawing

AI summary

A herbicidal composition comprisinga) at least one 3-phenyluracils of formula Iwherein the variables R1 to R7 are as defined in the specification; andb) at least one 3-sulfonylisoxazoline of formula IIwherein the variables R8 and R9 are as defined in the specification; andc) optionally at least one safener III selected from the group as defined in the specification.