Herbicidal Composition Synergy Reduces Application Rates

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Solution Overview

Problem

Current herbicide compositions face challenges in achieving effective weed control with lower application rates, often resulting in reduced selectivity and stability issues due to physical and biological incompatibilities between active compounds, which increases economic and environmental costs.

Innovation Solution

A composition combining herbicidally active compounds (A) and (B), where (A) represents compounds of a specific general formula or their agrochemically compatible salts, and (B) includes a range of herbicides from various groups, demonstrating synergistic effects that enhance activity and stability, allowing for reduced application rates and broader spectrum control.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If application rates of herbicides are increased to maintain efficacy, then weed control effectiveness is improved, but economic cost and environmental impact increase

Engineering Contradiction:
Improveweed control effectivenessVSAvoidapplication rate
Core Design Contradiction:
ReliabilityVSQuantity of substance

Solution Approach 1:

The patent combines compound (A) from formula (I) with compound (B) from formula (II) to create a synergistic herbicidal composition. This merging of two different herbicidal compounds produces an unexpected synergistic effect where the combination achieves superior weed control at lower application rates than either compound alone, thereby reducing both economic cost and environmental impact while maintaining or improving effectiveness

Inventive Principle:
Principle #5Merging (Combining)

2Adaptability or versatility

If multiple herbicides are combined to broaden spectrum control, then control of unwanted plant growth is improved, but physical and biological incompatibility increases

Engineering Contradiction:
Improvespectrum of controlVSAvoidstability of coformulation
Core Design Contradiction:
Adaptability or versatilityVSStability of the object's composition

Solution Approach 1:

The patent specifies precise structural parameters for compounds (A) and (B) including defined substituent groups (R1-R6, X1-X6, Z) and their possible variations. By controlling these chemical parameters and selecting specific combinations within defined ranges, the formulation achieves both broad spectrum control and stability, avoiding physical and biological incompatibility between the herbicides

Inventive Principle:
Principle #35Parameter changes

3Quantity of substance

If application rates are reduced to lower cost, then economic expenditure is reduced, but herbicidal action is insufficient

Engineering Contradiction:
Improveapplication rateVSAvoidherbicidal action
Core Design Contradiction:
Quantity of substanceVSReliability

Solution Approach 1:

The patent converts the potential harm of reduced application rates into a benefit by utilizing the synergistic interaction between compounds (A) and (B). The unexpected synergy means that lower doses of each compound, when combined, produce herbicidal action equal to or greater than higher doses of single compounds, thereby reducing cost while maintaining effectiveness

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

4Reliability

If higher application rates are used to compensate for resistance, then control of resistant harmful plants is improved, but selectivity of herbicides deteriorates

Engineering Contradiction:
Improvecontrol of resistant plantsVSAvoidselectivity
Core Design Contradiction:
ReliabilityVSObject-generated harmful factors

Solution Approach 1:

The patent creates a composite herbicidal system combining two chemically distinct compounds with different modes of action. This composite approach allows control of resistant weed populations through the combined effect of (A) and (B), while the specific structural definitions and synergistic interaction maintain selectivity, avoiding the need to increase application rates which would harm the crop

Inventive Principle:
Principle #40Composite materials

Data Source

PatentUS12171230B2Herbicidal compositions
Publication Date: 2024.12.24 BAYER AG
  • US12171230B2 patent drawing
  • US12171230B2 patent drawing
  • US12171230B2 patent drawing

AI summary

The present invention provides compositions comprising herbicidally active compounds (A) and (B), where (A) represents one or more compounds of the general formula (I) or their agrochemically acceptable salts [component (A)],and (B) represents one or more herbicides [component (B)]. The application furthermore relates to a method and to the use of the herbicidal composition according to the invention for controlling harmful plants or for regulating growth.