1,2-Hexanediol Stabilizes O/W Emulsions Against Phase Inversion

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Solution Overview

Problem

Oil-in-water emulsions with hydrophilic emulsifiers tend to experience phase inversion during production and storage, leading to instability, especially when using moderately polar to polar lipids with interfacial tension below 30 mN/m.

Innovation Solution

Incorporating 1,2-hexanediol in concentrations of 0.3% to 3% by weight and using oil-in-water emulsifiers like glyceryl stearate citrate, polyglyceryl methyl glucose distearate, and polyethylene glycol monostearate, along with additives such as tocopheryl acetate and phenoxyethanol, while maintaining a temperature between 30°C to 85°C during the emulsion production process.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If hydrophilic emulsifiers with HLB value ≥10 are used to produce O/W emulsions, then the emulsion can be formulated with water-soluble characteristics, but phase inversion occurs during production and storage leading to instability

Engineering Contradiction:
Improveemulsion formulation capabilityVSAvoidphase inversion resistance
Core Design Contradiction:
Adaptability or versatilityVSStability of the object's composition

Solution Approach 1:

The patent changes the chemical composition parameters of the oil phase by incorporating specific lipid types (neutral fats, fatty acid esters, triglycerides) with controlled interfacial tension properties. This parameter modification prevents phase inversion while maintaining the desired O/W emulsion structure and stability throughout storage.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite emulsion system combining hydrophilic emulsifiers with specifically selected lipid components. This composite approach synergistically prevents phase inversion by balancing the hydrophilic-lipophilic interactions, achieving both formulation flexibility and storage stability simultaneously.

Inventive Principle:
Principle #40Composite materials

2Ease of manufacture

If moderately polar to polar lipids with interfacial tension <30 mN/m are used in the oil phase, then the emulsion can be formulated with hydrophilic emulsifiers, but phase inversion tendency increases during storage

Engineering Contradiction:
Improveemulsion formulation easeVSAvoidstorage stability
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The patent modifies the interfacial tension parameter of the oil phase by selecting lipids with specific surface activity characteristics. This parameter adjustment allows the use of hydrophilic emulsifiers while preventing phase inversion during storage, achieving both ease of manufacture and storage reliability.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent introduces specific lipid components as intermediary substances that mediate between the hydrophilic emulsifier and the oil phase. These intermediary lipids with controlled interfacial tension properties prevent direct unfavorable interactions that would lead to phase inversion, maintaining stability throughout the product lifecycle.

Inventive Principle:
Principle #24Intermediary (Mediator)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The method significantly reduces phase inversion tendencies, resulting in a more stable cosmetic oil-in-water emulsion suitable for use as ointments, creams, or lotions, maintaining stability throughout storage.

Implementation Method 1

the problem often occurs that with the use of primarily moderately polar to polar lipids in the oil phase (i.e., lipids with a interfacial tension toward water of less than about 30 mN/m) an undesirable inversion of phases can occur. Furthermore, O/W emulsions of this type have a tendency towards phase inversion during storage

Methodology Applied
Scientific EffectPhase inversion prevention:

Implementation Method 2

Emulsifiers as a rule are molecules with a polar, hydrophilic structural element and a nonpolar, lipophilic structural element

Methodology Applied
Scientific EffectEmulsification: Emulsion

Implementation Method 3

lipids with a interfacial tension toward water of less than about 30 mN/m

Methodology Applied
Scientific EffectInterfacial tension reduction: Surface Tension

Implementation Method 4

one of the two liquids is dispersed in the form of very fine droplets in the other liquid. Outwardly and viewed with the naked eye, emulsions appear homogeneous

Methodology Applied
Scientific EffectDispersion: Dispersion (of waves)

Data Source

PatentUS8084507B2Cosmetic O/W emulsion comprising 1,2-hexanediol
Publication Date: 2011.12.27 BEIERSDORF AG

AI summary

A cosmetic oil-in-water emulsion which comprises 1,2-hexanediol and a method of preparing same.