HRV VLPs for Cross-Neutralizing Antibodies

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Solution Overview

Problem

Current vaccines fail to provide effective protection against the large number of human rhinovirus serotypes, as they do not induce a protective response that can cross-neutralize multiple serotypes, making it challenging to develop a vaccine that can protect against multiple HRV infections.

Innovation Solution

The development of virus-like particles (VLPs) comprising human rhinovirus capsid proteins VP0, VP1, and VP3, or VP1, VP2, and VP4, expressed as fusion proteins with SUMO sequences, which are used to induce an immune response and provide cross-neutralizing antibodies against multiple serotypes.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If traditional vaccines targeting single serotypes are used, then specific protection against that serotype is achieved, but protection against other serotypes is not provided

Engineering Contradiction:
Improveprotection efficacyVSAvoidcross-serotype coverage
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent employs conserved peptide sequences from multiple HRV serotypes (including clades A, B, and C) to create a vaccine composition that provides universal protection across different serotypes. The selected peptides from VP1, VP2, VP3, and VP4 proteins share high sequence identity across serotypes, enabling a single vaccine formulation to elicit cross-neutralizing antibodies against multiple HRV strains simultaneously.

Inventive Principle:
Principle #6Universality (Multi-functionality)

Solution Approach 2:

The vaccine composition combines multiple conserved peptide sequences from different viral proteins (VP1, VP2, VP3, VP4) and different serotypes into a composite formulation. This composite approach integrates epitopes from various viral components to generate a broader immune response that covers multiple serotypes, overcoming the limitation of single-serotype vaccines.

Inventive Principle:
Principle #40Composite materials

2Adaptability or versatility

If a vaccine targets multiple serotypes, then cross-protection is improved, but the complexity of identifying conserved regions across serotypes increases

Engineering Contradiction:
Improvecross-serotype coverageVSAvoidvaccine design complexity
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The patent divides the HRV capsid proteins into specific segmented regions (peptides of 6-20 amino acids) that exhibit conservation across serotypes. By focusing on discrete peptide segments from VP1, VP2, VP3, and VP4 proteins rather than entire proteins, the design process becomes more manageable while maintaining cross-serotype efficacy.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The vaccine design targets specific local regions (conserved peptide sequences) within the viral proteins that maintain high sequence identity across different serotypes. These localized conserved epitopes are selected based on their structural importance and conservation patterns, allowing focused vaccine development on critical regions rather than entire protein structures.

Inventive Principle:
Principle #3Local quality

3Reliability

If conserved peptides from multiple proteins are used, then cross-neutralizing activity is improved, but the manufacturing complexity increases

Engineering Contradiction:
Improvecross-neutralizing activityVSAvoidproduction simplicity
Core Design Contradiction:
ReliabilityVSEase of manufacture

Solution Approach 1:

The patent employs synthetic peptide sequences rather than requiring production of entire viral proteins or live attenuated viruses. These short conserved peptide sequences can be chemically synthesized using standard peptide synthesis methods, eliminating the need for complex cell culture systems, viral propagation, and extensive purification processes required for traditional vaccine platforms.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

Data Source

PatentEP3193922B1vaccine
Publication Date: 2019.08.28 GLAXOSMITHKLINE BIOLOGICALS SA
  • EP3193922B1 patent drawingFigure 1
  • EP3193922B1 patent drawingFigure 2
  • EP3193922B1 patent drawingFigure 3~4

AI summary

The present invention relates HRV VLPs and methods of making HRV VLPs.