HSV-NT3 Vector for Chemotherapy-Induced Peripheral Neuropathy

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Solution Overview

Problem

Chemotherapy-induced peripheral neuropathy (CIPN) is a debilitating side effect of cancer treatment that current treatments only partially address, with existing methods showing inconsistent success in managing symptoms and preventing nerve damage.

Innovation Solution

A herpes simplex virus (HSV) McKrae strain variant engineered to express neurotrophin 3 (NT3) is used, delivered via a viral vector that targets the dorsal root ganglia to provide prophylactic and therapeutic treatment, allowing for the prevention, inhibition, or reversal of neuropathy, enabling higher chemotherapy doses and longer treatment durations.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If chemotherapy is administered to treat cancer, then cancer treatment efficacy is improved, but chemotherapy-induced peripheral neuropathy (CIPN) occurs as a side effect

Engineering Contradiction:
Improvecancer treatment efficacyVSAvoidperipheral neuropathy
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent utilizes the HSV virus's natural tropism for neuronal cells and its ability to establish lifelong latency in the nervous system. By engineering the virus to express NT3 (a neuroprotective factor) instead of replicating, the harmful viral properties are converted into therapeutic benefit. The virus delivers neuroprotection precisely to the affected dorsal root ganglia where chemotherapy damage occurs, transforming a potential pathogen into a targeted delivery vehicle for neuropathy prevention and treatment.

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Solution Approach 2:

The HSV-NT3 vector serves as an intermediary between the chemotherapy treatment and the nervous system. It mediates protection by delivering NT3 directly to dorsal root ganglia, bridging the gap between systemic chemotherapy administration and localized neuroprotection. This intermediary approach allows high-dose chemotherapy to be administered while the vector simultaneously protects neural tissues from damage.

Inventive Principle:
Principle #24Intermediary (Mediator)

2Reliability

If higher chemotherapy doses are administered to improve treatment outcomes, then cancer treatment effectiveness increases, but neuropathy severity increases

Engineering Contradiction:
Improvecancer treatment effectivenessVSAvoidneuropathy severity
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The HSV-NT3 vector is administered before chemotherapy treatment begins, establishing neuroprotection in advance. The virus infects dorsal root ganglia and begins expressing NT3 prior to chemotherapy exposure, creating a protective environment that prevents neuropathy even when high-dose chemotherapy is subsequently administered. This preliminary action allows aggressive cancer regimens to proceed without neuropathy limitations.

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The invention changes the biochemical parameters within dorsal root ganglia by introducing NT3 expression. This alters the neurotrophic environment from one vulnerable to chemotherapy damage to one that is protected and supportive of neuronal survival. The parameter change in NT3 concentration enables tolerance to higher chemotherapy doses that would otherwise cause severe neuropathy.

Inventive Principle:
Principle #35Parameter changes

3Ease of operation

If existing neuropathy treatment methods are used, then some symptom relief is achieved, but treatment success is inconsistent and limited

Engineering Contradiction:
Improvesymptom managementVSAvoidtreatment success consistency
Core Design Contradiction:
Ease of operationVSReliability

Solution Approach 1:

The HSV-NT3 vector establishes self-sustaining neuroprotection that does not require repeated administrations or external intervention. Once the virus infects dorsal root ganglia, it maintains lifelong latency while continuously providing NT3 expression and neuroprotective effects. This self-service mechanism eliminates the inconsistency of current treatments that require frequent monitoring and adjustment, providing reliable, long-term protection.

Inventive Principle:
Principle #25Self-service

Solution Approach 2:

The vector provides continuous neuroprotection throughout the patient's life, unlike current treatments that are intermittent and short-term. The HSV maintains persistent latency in dorsal root ganglia, ensuring uninterrupted NT3 expression and ongoing protection against neuropathy. This continuity transforms neuropathy management from a series of discrete symptomatic interventions to a sustained protective therapy.

Inventive Principle:
Principle #20Continuity of useful action

Data Source

PatentEP3432905B1HSV vectors for delivery of NT3 and treatment of cipn
Publication Date: 2022.06.01 PERIPHAGEN INC
  • EP3432905B1 patent drawingFigure 1
  • EP3432905B1 patent drawingFigure 2
  • EP3432905B1 patent drawingFigure 3

AI summary

Disclosed herein are compositions and methods for treating neuropathy, embodiments, HSV vectors are provided comprising nucleic acid molecules encoding neurotrophins, such as neurotrophin 3 (NT3).