HYA Triglyceride Derivative for Liquid State and Flavor

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Solution Overview

Problem

10-hydroxy-cis-12-octadecenoic acid (HYA) has superior physiological functions but is solid at ambient temperature and has an acrid flavor, making it difficult to ingest and handle effectively.

Innovation Solution

A novel triglyceride is developed where at least one fatty acid forms an ester bond with the hydroxy group of glycerol, specifically using 10-hydroxy-cis-12-octadecenoic acid or its optical isomer, which is liquid at ambient temperature and has a good flavor, allowing for easy ingestion and handling.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If HYA is used directly, then physiological functions are improved, but handling and ingestion become difficult due to solid state and acrid flavor

Engineering Contradiction:
Improvephysiological functionVSAvoidhandling and ingestion
Core Design Contradiction:
ReliabilityVSEase of operation

Solution Approach 1:

The patent changes the physical state parameter of HYA from solid to liquid by converting it into a triglyceride derivative form. This parameter change resolves the contradiction by maintaining the physiological functionality of HYA while eliminating the handling difficulties associated with its solid state and acrid flavor.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite structure by incorporating HYA into a triglyceride molecule, where HYA forms an ester bond with glycerol. This composite approach allows HYA to be delivered in a form that combines the beneficial physiological effects of HYA with the favorable handling properties of liquid triglycerides.

Inventive Principle:
Principle #40Composite materials

2Ease of operation

If HYA is converted to triglyceride derivative, then handling and ingestion become easy, but the direct physiological effect may be reduced

Engineering Contradiction:
Improvehandling and ingestionVSAvoidphysiological function
Core Design Contradiction:
Ease of operationVSReliability

Solution Approach 1:

The triglyceride derivative acts as an intermediary carrier that delivers HYA to the body. The ester bond in the triglyceride structure allows for enzymatic hydrolysis in the digestive system, releasing free HYA that can then exert its physiological effects. This intermediary approach resolves the contradiction by facilitating easy ingestion while ensuring physiological functionality is restored through in vivo hydrolysis.

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent performs preliminary action by pre-converting HYA into a triglyceride derivative form that is easier to handle and ingest. This preliminary transformation does not permanently alter HYA's functionality, as the ester bond can be broken down in the body to release the active HYA molecule when needed.

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The triglyceride derivative is liquid at ambient temperature, has a pleasant flavor, and upon ingestion, the ester bond is hydrolyzed by lipase, releasing HYA, thereby exerting its superior physiological functions such as improving lipid metabolism and enhancing intestinal immunity.

Implementation Method 1

the ester bond is hydrolyzed by lipase, releasing HYA

Methodology Applied
Scientific EffectHydrolysis: Hydrolysis

Data Source

PatentEP3305756B1Novel triglyceride and use thereof
Publication Date: 2022.01.05 NOSTER INC
  • EP3305756B1 patent drawingFigure 1
  • EP3305756B1 patent drawingFigure 2
  • EP3305756B1 patent drawingFigure 3-1

AI summary

The present invention provides a novel HYA derivative having superior physiological functions intrinsic to HYA and permitting easy ingestion and easy handling, and use thereof. The present invention relates to a triglyceride in which at least one fatty acid forming an ester bond with a hydroxy group of glycerol is 10-hydroxy-cis-12-octadecenoic acid, or an optical isomer thereof, and a composition (edible fat or oil, food, medicament, cosmetic etc.) containing same.