Implantable Microneedle Patch with Dissolvable Base

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Solution Overview

Problem

Current microneedle technologies face challenges in achieving sufficient mechanical strength and controlled drug release, often requiring complex manufacturing processes and high costs, while also struggling with the need for long-term application to ensure sustained release.

Innovation Solution

The development of an implantable sustained-release microneedle patch using a polylactic acid-based needle tip center layer and a water-soluble polymer material for the needle body, base, and outer layer, which enhances mechanical strength and skin penetration, allowing for efficient drug delivery and prolonged release without the need for long-term application.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Strength

If traditional metal, glass, or silicon microneedles are used, then mechanical strength is improved, but safety deteriorates due to breaking and leaving residues in the skin

Engineering Contradiction:
Improvemechanical strengthVSAvoidsafety
Core Design Contradiction:
StrengthVSObject-affected harmful factors

Solution Approach 1:

The patent changes the material parameter from traditional metal/glass/silicon to biodegradable polymer materials (PLA, PGA, PLGA) that maintain sufficient mechanical strength for skin penetration while eliminating the harmful effect of breaking and leaving residues. The polymer materials are specifically selected to degrade safely in the body over time.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent employs composite material structures combining biodegradable polymer matrices with embedded drug particles or microsphere carriers. This composite approach allows the microneedle to achieve both mechanical strength for penetration and controlled drug release functionality, while the polymer matrix ensures safe biodegradation without harmful residues.

Inventive Principle:
Principle #40Composite materials

2Object-affected harmful factors

If polymer microneedles with water-soluble or biodegradable materials are used, then safety is improved, but manufacturing complexity increases due to specific material requirements

Engineering Contradiction:
ImprovesafetyVSAvoidmanufacturing complexity
Core Design Contradiction:
Object-affected harmful factorsVSDevice complexity

Solution Approach 1:

The patent simplifies manufacturing by selecting polymer materials with appropriate melting points and processing characteristics. The biodegradable polymers are chosen to be processable using conventional microneedle manufacturing techniques, avoiding the need for complex specialized equipment while maintaining safety benefits.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent utilizes biodegradable polymer materials that can be easily manufactured and disposed of after serving their purpose. The materials are designed to degrade in the body after delivering the drug payload, eliminating the need for complex retrieval mechanisms and simplifying both manufacturing and clinical application.

Inventive Principle:
Principle #27Cheap short-living objects (Disposable)

3Duration of action of moving object

If microneedles are designed for sustained-release, then duration of action is improved, but device complexity increases due to controlled release mechanisms

Engineering Contradiction:
Improveduration of actionVSAvoiddevice complexity
Core Design Contradiction:
Duration of action of moving objectVSDevice complexity

Solution Approach 1:

The patent incorporates drug-loaded microsphere carriers or particles during the microneedle manufacturing process, so that the controlled release mechanism is pre-established within the microneedle structure. This preliminary action allows sustained-release functionality to be built-in without adding complex external control mechanisms.

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The patent employs biodegradable polymer matrices that automatically control drug release through their natural degradation process. The microneedle structure itself serves as the release mechanism, with the polymer degrading over time to release the embedded drug payload without requiring external control systems or additional complexity.

Inventive Principle:
Principle #25Self-service

4Duration of action of moving object

If microneedles require long-term application for sustained release, then duration of action is improved, but loss of time increases due to extended application period

Engineering Contradiction:
Improveduration of actionVSAvoidapplication time
Core Design Contradiction:
Duration of action of moving objectVSLoss of time

Solution Approach 1:

The patent loads drugs into the microneedle structure during manufacturing, with the biodegradable polymer matrix designed to release the drug over a controlled period. This preliminary loading allows the microneedle to provide sustained release functionality without requiring prolonged application time from the user, as the release mechanism is activated upon insertion and degrades automatically.

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

This solution provides a microneedle patch with improved mechanical strength and skin penetration, enabling efficient drug delivery and prolonged release, reducing manufacturing complexity and cost, and eliminating the need for long-term application.

Implementation Method 1

the needle tip and the needle body and the base are formed of different matrices; the needle body and the base being formed of a matrix comprising a water-soluble polymer material... the needle tip will be separated from the needle body and the base

Methodology Applied
Scientific EffectDissolution: Solvation

Implementation Method 2

the needle tip center layer is formed of a matrix comprising a biodegradable water-insoluble polymer material... achieving purposes of convenience, safety, biodegradability, and efficient administration

Methodology Applied
Scientific EffectHydrolysis: Hydrolysis

Data Source

PatentEP3845216B1Implantable sustained-release microneedle patch and preparation method therefor
Publication Date: 2025.04.09 BEIJING CAS MICRONEEDLE TECH LTD
  • EP3845216B1 patent drawingFigure 1~2
  • EP3845216B1 patent drawingFigure 3~4
  • EP3845216B1 patent drawingFigure 5~7

AI summary

An implantable sustained-release microneedle patch and a preparation method therefor. The implantable sustained-release microneedle comprises a needle tip, a needle body, and a base. The needle tip comprises a needle tip center layer and a needle tip outer layer. The needle tip center layer is formed of a matrix comprising a biodegradable water-insoluble polymer material. The needle tip outer layer, the needle body, and the base are formed of a matrix comprising a water-soluble polymer material. The microneedle patch comprises the microneedle and absorbs the moisture of the skin when the microneedle acts on skin, so that the base and the needle body are quickly separated from the needle tip within 0.5-2 h. After the base is removed, the needle tip will be left in skin, and the user does not need the patch sticking for a long time to ensure long-term release of a drug in the body.