Quick Release Insecticidal Granules via Surfactant Carrier Matrix

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Solution Overview

Problem

Current agrochemical formulations, particularly granular formulations containing chlorantraniliprole, face challenges in achieving quick and efficient release of active ingredients, leading to inadequate pest control and potential environmental concerns due to excessive active ingredient amounts and resistance issues.

Innovation Solution

A quick release insecticidal composition comprising a diamide insecticide like chlorantraniliprole, dispersed in a carrier matrix comprising a binder and a surfactant, which facilitates rapid release upon contact with water, ensuring effective pest control with controlled active ingredient distribution.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Speed

If active ingredients are formulated with inert ingredients in granular formulations, then the desired dosage form and characteristics are obtained, but the active ingredients are not released to their full extent in the required time

Engineering Contradiction:
Improverelease rate of active ingredientVSAvoidpest control effectiveness
Core Design Contradiction:
SpeedVSReliability

Solution Approach 1:

The patent changes the chemical and physical parameters of the carrier matrix by incorporating specific surfactants (anionic, cationic, nonionic, or amphoteric) and binders in optimized ratios. This modifies the matrix properties to enable rapid dissolution and release of chlorantraniliprole, achieving over 60% release within 1 hour while maintaining formulation stability and pest control effectiveness

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates a composite carrier matrix system combining multiple components: binders (natural or synthetic polymers), surfactants (various types), and inert ingredients. This composite structure facilitates both the mechanical integrity of granules and the rapid release of active ingredient through synergistic interactions among components

Inventive Principle:
Principle #40Composite materials

2Reliability

If greater amounts of active ingredient are used, then pest control is improved, but environmental leaching risk and economic cost increase

Engineering Contradiction:
Improvepest control effectivenessVSAvoidenvironmental leaching risk
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent designs a controlled release system where the carrier matrix continuously releases active ingredient over time, maintaining effective concentrations at the pest site. This continuous release mechanism ensures sustained pest control with smaller total amounts of active ingredient, reducing environmental leaching while maintaining reliability

Inventive Principle:
Principle #20Continuity of useful action

Solution Approach 2:

The carrier matrix acts as an intermediary between the active ingredient and the environment, controlling the release kinetics and preventing premature leaching. The matrix components (binders, surfactants) mediate the release process, ensuring active ingredient is delivered efficiently to target pests rather than leaching into environment

Inventive Principle:
Principle #24Intermediary (Mediator)

3Object-affected harmful factors

If smaller amounts of active ingredient are used, then environmental and economic concerns are reduced, but pest control effectiveness decreases and resistance risk increases

Engineering Contradiction:
Improveenvironmental and economic impactVSAvoidpest control effectiveness
Core Design Contradiction:
Object-affected harmful factorsVSReliability

Solution Approach 1:

The patent optimizes formulation parameters including surfactant concentration (0.1-30% w/w), binder ratio (1:5 to 5:1), and active ingredient content (0.1-70% w/w) to maximize release efficiency. These parameter changes enable smaller amounts of active ingredient to achieve equivalent pest control by improving bioavailability and release kinetics

Inventive Principle:
Principle #35Parameter changes

4Ease of operation

If chlorantraniliprole is formulated in water-based granular system, then ease of application is improved, but the poor water solubility of chlorantraniliprole makes ready availability difficult

Engineering Contradiction:
Improveease of application in water-based systemVSAvoidrelease rate of active ingredient
Core Design Contradiction:
Ease of operationVSSpeed

Solution Approach 1:

The patent uses surfactants as intermediary substances that bridge the hydrophobic chlorantraniliprole and the aqueous environment. These surfactants form micelles or complexes with the active ingredient, enabling its dissolution and dispersion in water-based granular formulations while maintaining rapid release capability

Inventive Principle:
Principle #24Intermediary (Mediator)

Solution Approach 2:

The patent modifies the solubility parameters of chlorantraniliprole by incorporating surfactants that change the physical-chemical environment. The surfactant molecules interact with the hydrophobic active ingredient, effectively increasing its apparent water solubility and enabling ready availability in water-based systems

Inventive Principle:
Principle #35Parameter changes

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The composition achieves rapid release of at least 60% of the active ingredient within 1 hour, enhancing pest control efficacy while minimizing environmental impact and reducing resistance risks.

Implementation Method 1

a carrier matrix comprising a binder and a surfactant, wherein the diamide insecticide is dispersed in the carrier matrix

Methodology Applied
Scientific EffectSurfactant action: Surfactant

Implementation Method 2

a carrier matrix comprising a binder and a surfactant

Methodology Applied
Scientific EffectBinding: Binder

Data Source

PatentUS20240000072A1Quick release insecticidal composition
Publication Date: 2024.01.04 UPL LTD

AI summary

A quick release insecticidal composition is provided. Also provided is a process of preparing a quick release insecticidal composition. Methods of controlling pests comprising applying the quick release insecticidal composition to a pest or to a locus comprising the pest are also disclosed.