Intestinal Bacterial Composition to Block Drug-Resistant Colonization

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Solution Overview

Problem

There is a need for an effective antibacterial composition that can suppress the colonization and proliferation of drug-resistant bacteria and pro-inflammatory bacteria in the intestinal tract, which are associated with various diseases.

Innovation Solution

The development of an antibacterial composition containing specific intestinal bacteria strains, such as those identified by their 16S rDNA sequences, which can suppress the colonization of drug-resistant bacteria and pro-inflammatory bacteria, including strains like Kp2H7, by administering these strains to the intestinal tract.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Ease of operation

If antibiotic administration is performed to eliminate intestinal bacteria, then the intestinal tract becomes available for colonization by Th1 cell-inducible bacteria, but this leads to increased colonization of drug-resistant bacteria and pro-inflammatory bacteria

Engineering Contradiction:
Improveavailability of intestinal tract for colonizationVSAvoidcolonization of drug-resistant bacteria
Core Design Contradiction:
Ease of operationVSObject-affected harmful factors

Solution Approach 1:

The patent applies preliminary anti-action by administering beneficial intestinal bacteria (such as Lactobacillus, Bifidobacterium, or other probiotic strains) before or concurrently with antibiotic treatment. These beneficial bacteria preemptively occupy ecological niches in the intestinal tract, preventing drug-resistant bacteria and pro-inflammatory bacteria from colonizing even when antibiotics eliminate the normal flora. This is demonstrated in the examples where probiotic administration suppressed the colonization of pathogenic bacteria despite antibiotic-induced flora disruption

Inventive Principle:
Principle #9Preliminary anti-action

Solution Approach 2:

The patent uses beneficial intestinal bacteria as an intermediary organism that mediates between the antibiotic treatment and the pathogenic bacteria. These intermediary bacteria interact with the intestinal environment and pathogenic organisms through competitive exclusion, production of antimicrobial substances, and modulation of the immune response, thereby preventing direct colonization of harmful bacteria while allowing the antibiotic therapy to proceed

Inventive Principle:
Principle #24Intermediary (Mediator)

2Adaptability or versatility

If oral bacteria colonize in the intestinal tract, then Th1 cells are induced and proliferate, but this leads to development of diseases such as Crohn's disease, liver cirrhosis, and colorectal cancer

Engineering Contradiction:
Improvecolonization capability of oral bacteriaVSAvoiddisease development
Core Design Contradiction:
Adaptability or versatilityVSObject-generated harmful factors

Solution Approach 1:

The patent applies preliminary anti-action by introducing beneficial intestinal bacteria that preemptively prevent oral bacteria from colonizing the intestinal tract. These beneficial bacteria establish themselves in the intestinal ecosystem first, creating a protective barrier that blocks the colonization of Th1 cell-inducible oral bacteria, thereby preventing the downstream inflammatory response and disease development associated with such colonization

Inventive Principle:
Principle #9Preliminary anti-action

Solution Approach 2:

The patent converts the potential harm of bacterial colonization into a benefit by using beneficial bacteria to occupy the ecological niche that would otherwise be taken by harmful oral bacteria. The same colonization mechanism that causes disease when performed by oral bacteria is harnessed for protection when performed by probiotic strains, transforming the colonizable state of the intestinal tract from a vulnerability into a defense mechanism

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

3Ease of manufacture

If intestinal bacteria are eliminated by antibiotic administration, then the intestinal flora is disrupted, but this creates an opportunity for drug-resistant bacteria to colonize and proliferate

Engineering Contradiction:
Improveelimination of competing intestinal bacteriaVSAvoidsuppression of drug-resistant bacteria
Core Design Contradiction:
Ease of manufactureVSReliability

Solution Approach 1:

The patent applies preliminary anti-action by administering probiotic bacteria before or during antibiotic treatment to preemptively block the colonization of drug-resistant bacteria. While antibiotics eliminate competing intestinal bacteria, the probiotics are either resistant to the antibiotics or are administered in sufficient quantities to repopulate the intestinal tract rapidly, maintaining suppression of drug-resistant organisms throughout the treatment period

Inventive Principle:
Principle #9Preliminary anti-action

Solution Approach 2:

The patent applies preliminary action by pre-establishing a population of beneficial bacteria in the intestinal tract before antibiotic administration begins. This preliminary colonization ensures that when antibiotics disrupt the normal flora, the probiotic bacteria are already in position to prevent drug-resistant bacteria from establishing themselves, maintaining reliable suppression throughout the antibiotic treatment course

Inventive Principle:
Principle #10Preliminary action

Data Source

PatentEP3957367B1Antibacterial composition against drug-resistant bacteria or pro-inflammatory bacteria
Publication Date: 2026.01.14 KEIO UNIV
  • EP3957367B1 patent drawingFigure 1
  • EP3957367B1 patent drawingFigure 2
  • EP3957367B1 patent drawingFigure 3

AI summary

The present invention provides an antibacterial composition against drug-resistant bacteria or pro-inflammatory bacteria containing an intestinal bacterium as an active ingredient, or a pharmaceutical composition for treating, ameliorating, or preventing an infectious disease or an inflammatory disease.