Lixisenatide Glycemic Control in Pediatric Type 2 Diabetes

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Solution Overview

Problem

Current treatments for type 2 diabetes mellitus in pediatric patients, particularly those with high body mass index (BMI) ≥ 30 kg/m², often fail to adequately control blood glucose levels, leading to increased risks of cardiovascular diseases and diabetes complications due to insufficient glycemic control, especially when metformin monotherapy or basal insulin therapy is insufficient.

Innovation Solution

The use of lixisenatide, a GLP-1 analogue, either alone or in combination with metformin and/or basal insulin, to improve glycemic control in pediatric patients with type 2 diabetes mellitus, as it reduces postprandial plasma glucose, insulin, and glucagon secretion, thereby achieving better glucose regulation.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If metformin monotherapy or basal insulin therapy is used in pediatric patients with high BMI, then treatment simplicity is maintained, but glycemic control becomes insufficient

Engineering Contradiction:
Improveglycemic controlVSAvoidtreatment regimen
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent combines lixisenatide with metformin and/or basal insulin to create a multi-component therapeutic regimen. This merging of treatments addresses the insufficiency of monotherapy while managing the complexity through structured combination protocols for pediatric patients with high BMI and inadequate glycemic control

Inventive Principle:
Principle #5Merging (Combining)

2Reliability

If conventional treatments are used in pediatric patients with type 2 diabetes, then treatment accessibility is maintained, but diabetes complications increase due to insufficient glycemic control

Engineering Contradiction:
Improveglycemic controlVSAvoiddiabetes complications
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent applies preliminary anti-action by using lixisenatide to proactively reduce postprandial glucose excursions and suppress glucagon secretion before hyperglycemia can lead to complications. This preventive approach targets the underlying mechanisms of glucose dysregulation in pediatric type 2 diabetes to prevent future complications

Inventive Principle:
Principle #9Preliminary anti-action

3Reliability

If lixisenatide is added to improve glycemic control, then glycemic control improves, but treatment complexity increases

Engineering Contradiction:
Improveglycemic controlVSAvoidtreatment regimen
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent implements a dynamic treatment approach where lixisenatide is added based on specific clinical criteria (BMI ≥30 kg/m² and inadequate control on metformin and/or basal insulin). The treatment regimen can be adjusted by modifying lixisenatide dosage or discontinuing based on glycemic control response, allowing flexibility to balance efficacy with treatment complexity

Inventive Principle:
Principle #15Dynamics

Data Source

PatentEP3244912B1Treatment of pediatric type 2 diabetes mellitus patients with lixisenatide
Publication Date: 2021.08.18 SANOFI AVENTIS DEUT GMBH
  • EP3244912B1 patent drawingFigure 1~2
  • EP3244912B1 patent drawingFigure 3
  • EP3244912B1 patent drawingFigure 4

AI summary

The present invention refers to lixisenatide for use in pediatrics.