M13 Phage Display Vectors for Longer Peptide Integration

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Solution Overview

Problem

Current phage display systems using type 33 vectors face limitations in displaying longer peptides, as they reduce phage infectivity and result in lower copy numbers, making it difficult to isolate target-specific peptides with high affinity.

Innovation Solution

Introducing defined mutations in the wild-type g.III gene of type 33 bacteriophage M13 vectors to reduce the incorporation of the polypeptide encoded by the mutated gene, thereby increasing the display of exogenous peptides up to 35 amino acids on the phage surface while maintaining phage infectivity.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If type 33 vectors are used to display longer peptides, then peptide display capability is improved, but phage infectivity is reduced

Engineering Contradiction:
Improvepeptide display capabilityVSAvoidphage infectivity
Core Design Contradiction:
Adaptability or versatilityVSReliability

Solution Approach 1:

The patent applies parameter changes by modifying the signal peptide sequence parameters (amino acid composition, charge distribution, hydrophobicity) to optimize the balance between peptide display capability and phage infectivity. Specific substitutions in the signal peptide sequence alter its processing efficiency and routing, enabling longer peptides to be displayed while maintaining adequate infectivity levels.

Inventive Principle:
Principle #35Parameter changes

2Quantity of substance

If type 3 vectors are used to display peptides, then display copy number is increased, but peptide length is limited

Engineering Contradiction:
Improvedisplay copy numberVSAvoidpeptide length
Core Design Contradiction:
Quantity of substanceVSLength of moving object

Solution Approach 1:

The patent applies segmentation by dividing the single g.III gene into two separate copies (g.IIIa and g.IIIb), each capable of independent expression. This allows the system to accommodate longer peptide sequences that would be too bulky for a single gene product, while still achieving sufficient display copy numbers through the combined contribution of both gene copies.

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The patent modifies parameters of the g.III gene copies, including signal peptide sequences and coding regions, to optimize their expression levels and functional properties. These parameter changes enable each copy to contribute effectively to peptide display while accommodating longer peptide sequences.

Inventive Principle:
Principle #35Parameter changes

3Productivity

If wild-type g.III gene is used, then phage assembly is efficient, but exogenous peptide display is limited

Engineering Contradiction:
Improvephage assembly efficiencyVSAvoidexogenous peptide display
Core Design Contradiction:
ProductivityVSAdaptability or versatility

Solution Approach 1:

The patent applies local quality by making specific localized modifications to the g.III gene sequence while preserving the overall structure and function necessary for phage assembly. The modifications are concentrated in specific regions (signal peptide, coding sequence) that control peptide display, while the rest of the protein maintains its native assembly function.

Inventive Principle:
Principle #3Local quality

Solution Approach 2:

The patent changes parameters of the g.III gene including signal peptide sequence composition, coding region length, and amino acid composition to enable exogenous peptide display. These parameter changes are optimized to maintain sufficient phage assembly efficiency while providing the necessary capacity for displaying modified or longer peptide sequences.

Inventive Principle:
Principle #35Parameter changes

Data Source

PatentUS11066460B2Phage display vectors and methods of use
Publication Date: 2021.07.20 ELI LILLY & CO

AI summary

The present invention relates to vectors suitable for use in displaying proteins on the surface of bacteriophage M13 as fusion constructs with the surface protein P.III, bacteriophage M13 particles comprising a mutated P.III protein on the phage coat surface, as well as methods for producing bacteriophage M13 particles and methods for transfecting or infecting a host cell comprising the vectors and bacteriophage of the invention.