Mectin Nanoparticle Formulations for Soil Mobility

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Solution Overview

Problem

Mectin and milbemycin insecticides face challenges due to rapid degradation, poor water solubility, and lack of systemic activity, leading to frequent applications and reduced efficacy in agricultural use.

Innovation Solution

Formulations of nanoparticles of polymer-associated mectin or milbemycin compounds with specific formulating agents, such as polyelectrolytes and dispersants, are developed to enhance stability, solubility, and mobility, allowing for improved application and pest control.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If traditional mectin and milbemycin formulations are used, then pest control activity is achieved, but rapid degradation and photolysis reduce stability and duration of action

Engineering Contradiction:
ImprovestabilityVSAvoidduration of action
Core Design Contradiction:
ReliabilityVSDuration of action of stationary object

Solution Approach 1:

The patent segments the active ingredient into nanoparticle formulations (1-1000 nm), dividing the bulk chemical into controlled-release particles that degrade more slowly and provide sustained pest control activity over extended periods

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The active ingredient is nested within polymer matrices and encapsulated in nanoparticle structures, providing protective layers that shield against photolysis and degradation while enabling controlled release over time

Inventive Principle:
Principle #7Nested doll (Nesting)

2Reliability

If traditional formulations are applied, then some pest control is achieved, but poor water solubility limits mobility and distribution in soil

Engineering Contradiction:
ImproveefficacyVSAvoidmobility
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent changes the physical parameters of the formulation by creating nanoparticles with specific size distributions (1-1000 nm) and using polymer associations that enhance water solubility while maintaining soil mobility and distribution capabilities

Inventive Principle:
Principle #35Parameter changes

3Duration of action of stationary object

If macrocyclic lactones are taken up by plant leaves, then residual activity against mites is demonstrated, but lack of phloem and xylem mobility prevents true systemic effect

Engineering Contradiction:
Improveresidual activityVSAvoidsystemic effect
Core Design Contradiction:
Duration of action of stationary objectVSAdaptability or versatility

Solution Approach 1:

The patent transitions from foliar application with limited translocation to root-directed nanoparticle formulations that exploit the nanoparticle size advantage to achieve systemic movement through soil and plant uptake pathways, adding a new dimension of delivery

Inventive Principle:
Principle #17Another dimension (Dimensionality change)

4Reliability

If frequent applications are made to compensate for rapid degradation, then pest control is maintained, but application frequency increases and efficiency decreases

Engineering Contradiction:
Improvepest controlVSAvoidapplication efficiency
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The nanoparticle formulations provide continuous release of the active ingredient over extended periods, maintaining effective concentrations for pest control without requiring frequent reapplication, thus improving application efficiency

Inventive Principle:
Principle #20Continuity of useful action

Data Source

PatentUS9961901B2Mectin and milbemycin nanoparticle formulations
Publication Date: 2018.05.08 VIVE CROP PROTECTION INC

AI summary

The present disclosure describes a formulation including a nanoparticle including a polymer-associated mectin and/or milbemycin compounds with an average diameter of between about 1 nm and about 500 nm; wherein the polymer is a polyelectrolyte, and a dispersant or a wetting agent. The disclosure describes various formulations and formulating agents that can be included in the formulations. Additionally, the disclosure describes application to various plants and pests as well as advantages of the disclosed formulations.