Synergistic Microbicidal Composition for Resistant Strains

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Solution Overview

Problem

Commercial microbicides often fail to provide effective control of microorganisms, especially resistant strains and in aggressive environmental conditions, necessitating the development of synergistic combinations for enhanced activity at lower concentrations for economic and environmental benefits.

Innovation Solution

A microbicidal composition comprising 1,2-benzisothiazolin-3-one and various microbicides such as benzalkonium chloride, benzethonium chloride, or 2-methyl-4-isothiazolin-3-one with caprylyl glycol, which together exhibit enhanced efficacy at lower combined active ingredient levels, providing effective control of microorganisms.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If higher concentrations of individual microbicides are used, then microbicidal activity is improved, but environmental harm and cost increase

Engineering Contradiction:
Improvemicrobicidal activityVSAvoidenvironmental harm
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent combines multiple microbicides (1,2-benzisothiazolin-3-one with benzalkonium chloride, benzethonium chloride, or 2-methyl-4-isothiazolin-3-one with caprylyl glycol) to create synergistic formulations. This merging of substances achieves enhanced microbicidal activity at lower overall concentrations, thereby maintaining effectiveness while reducing environmental harm and cost associated with using high concentrations of single microbicides.

Inventive Principle:
Principle #5Merging (Combining)

2Reliability

If higher concentrations of individual microbicides are used, then microbicidal activity is improved, but cost increases

Engineering Contradiction:
Improvemicrobicidal activityVSAvoidcost
Core Design Contradiction:
ReliabilityVSQuantity of substance

Solution Approach 1:

The patent combines multiple microbicides to create synergistic formulations that achieve enhanced microbicidal activity at lower overall concentrations. This merging approach reduces the total quantity of active ingredients needed, thereby lowering cost while maintaining or improving microbicidal activity compared to using higher concentrations of single microbicides.

Inventive Principle:
Principle #5Merging (Combining)

3Device complexity

If single microbicides are used, then formulation simplicity is maintained, but effectiveness against resistant strains decreases

Engineering Contradiction:
Improveformulation simplicityVSAvoideffectiveness against resistant strains
Core Design Contradiction:
Device complexityVSReliability

Solution Approach 1:

The patent combines multiple microbicides with different mechanisms of action to create formulations that are effective against resistant microbial strains. The synergistic combination of 1,2-benzisothiazolin-3-one with benzalkonium chloride or benzethonium chloride, and 2-methyl-4-isothiazolin-3-one with caprylyl glycol, provides broad-spectrum activity that overcomes resistance while maintaining reasonable formulation simplicity.

Inventive Principle:
Principle #5Merging (Combining)

Data Source

PatentUS7468384B2Microbicidal composition
Publication Date: 2008.12.23 NUTRITION & BIOSCIENCES USA 2 LLC

AI summary

A microbicidal composition of 1,2-benzisothiazolin-3-one; and at least one of benzalkonium chloride, benzethonium chloride, benzyl alcohol, caprylyl glycol, chlorphenesin, diazolidinyl urea, ethylparaben, imidazolidinyl urea, methylparaben, phenoxyethanol, linoleamidopropyl PG-dimonium chloride phosphate, cocamidopropyl PG-dimonium chloride phosphate, propylparaben, cis-1-(3-chloroallyl)-3,5,7-triaza-1-azoniaadamantane chloride, dehydroacetic acid or its salts, benzoic acid or its salts, and sodium hydroxymethylglycinate.