Modified PFK Enzyme Enables Pentose Fermentation in Yeast

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Solution Overview

Problem

Current methods for bio-ethanol production from lignocellulose materials are hindered by Saccharomyces cerevisiae's inability to efficiently ferment pentose sugars due to low expression levels of key enzymes and redox imbalance, limiting productivity and yield.

Innovation Solution

Modification of the glycolytic enzyme 6-phosphofructo-1-kinase (PFK) to form active shorter fragments, combined with expression of a NADPH-specific malic enzyme, enables recombinant yeast cells to ferment pentose sugars and produce fermentative products like 2-phenylethanol by optimizing metabolic flux and redox balance.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If Saccharomyces cerevisiae is used for bio-ethanol production, then ethanol tolerance and accumulation yield are improved, but the ability to ferment pentose sugars is lost

Engineering Contradiction:
Improveethanol toleranceVSAvoidpentose sugar fermentation ability
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent divides the complex metabolic pathway into separate functional modules: introducing heterologous xylose utilization genes (xylA, xylB, xylC from P. stipitis) while maintaining the native S. cerevisiae ethanol production pathway. This segmentation allows the yeast to acquire pentose fermentation capability without losing its superior ethanol tolerance, as each pathway operates semi-independently within the cell

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

The modified S. cerevisiae strain achieves multi-functionality by combining native glucose fermentation and ethanol production capabilities with newly acquired xylose and arabinose utilization pathways. The yeast becomes a universal platform that can process multiple sugar types (glucose, xylose, arabinose) while maintaining high ethanol tolerance, effectively serving multiple functions in bio-ethanol production from lignocellulose

Inventive Principle:
Principle #6Universality (Multi-functionality)

2Adaptability or versatility

If heterologous genes for pentose sugar degradation are inserted, then pentose fermentation capability is improved, but gene expression levels and metabolic flux remain insufficient

Engineering Contradiction:
Improvepentose sugar fermentation capabilityVSAvoidmetabolic flux
Core Design Contradiction:
Adaptability or versatilityVSProductivity

Solution Approach 1:

The patent employs parameter changes by using strong constitutive promoters (GPD, GAPDH, TEF1) to drive high-level expression of heterologous xylose utilization genes. This ensures that the introduced genes are expressed at sufficient levels to achieve meaningful metabolic flux through the pentose degradation pathway, transforming the low-expression state into a high-flux state capable of supporting viable pentose fermentation

Inventive Principle:
Principle #35Parameter changes

3Productivity

If xylose utilization genes are overexpressed, then pentose assimilation is improved, but redox balance (NADH/NADPH ratio) becomes unbalanced

Engineering Contradiction:
Improvexylose assimilation rateVSAvoidredox balance
Core Design Contradiction:
ProductivityVSStability of the object's composition

Solution Approach 1:

The patent implements metabolic feedback balance by carefully selecting and coordinating the expression of multiple enzymes in the xylose utilization pathway. The xylA (xylose reductase), xylB (xylitol dehydrogenase), and xylC (xylulokinase) genes are co-expressed with balanced promoter strengths, creating a feedback-regulated system that maintains NADH/NADPH homeostasis while achieving high xylose assimilation rates

Inventive Principle:
Principle #23Feedback

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The modified PFK and malic enzyme system allows for efficient growth on pentose sugars and increased production of fermentative products, such as 2-phenylethanol, under semi-anaerobic conditions, enhancing bio-ethanol production and metabolic efficiency.

Implementation Method 1

a modified glycolytic enzyme 6-phosphofructo-1-kinase (PFK) that enables fermentative growth

Methodology Applied
Scientific EffectEnzyme catalysis: Enzyme

Implementation Method 2

expression of a NADPH-specific malic enzyme, enables recombinant yeast cells to ferment pentose sugars

Methodology Applied
Scientific EffectRedox reaction: Redox Reactions

Implementation Method 3

enables fermentative growth of the recombinant yeast Saccharomyces cerevisiae cells on pentose sugars

Methodology Applied
Scientific EffectFermentation: Fermentation

Data Source

PatentEP3274449B1Modified 6-phosphofructo-1 -kinases, which enable frementative growth of recombinant yeast saccharomyces cerevisiae cells on pentose sugars
Publication Date: 2020.03.04 KEMIJSKI INST
  • EP3274449B1 patent drawingFigure 1a~1b
  • EP3274449B1 patent drawingFigure 2~3
  • EP3274449B1 patent drawingFigure 4~5

AI summary

The subject of the invention is the modified glycolytic enzyme 6-phosphofructo-1 -kinase (PFK) that will allow the yeast Saccharomyces cerevisiae cells to fermentatively grow on pentose sugars. The invention belongs to the field of genetic engineering and microbial cells and fermentations or processes for the synthesis of desired chemical compounds, more specifically into the field of fermentative products formation that are based on the expression of the modified genes in the host cell. The essence of the invention is a modification of the gene encoding 6-phosphofructo-1- kinase (PFK), the key regulatory enzyme, of glycolysis that determines the rate of metabolic flux through the initial part of primary metabolism. Modified gene is of human, animal, microbial origin or it is a hybrid. A consequence of modified pfk genes expression in a host cell is the formation of the shorter PFK fragments that have higher activities in respect to the native enzyme. Modified enzymes in combination with NADPH-specific malic enzyme enable the use of pentose sugars and production of fermentative products, in particular 2-phenyethanol.