Multi-substituted Hydroxyapatite Bone Substitute

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Solution Overview

Problem

Current bone substitutes made from stoichiometric hydroxyapatite are not biocompatible and biomimetic enough to effectively integrate and replace natural bone tissue, leading to slow integration and regeneration times due to insufficient osteoblast activation and reabsorbability issues.

Innovation Solution

Development of hydroxyapatite multi-substituted with Sr2+ ions and optionally silicate and/or carbonate ions, optimized to achieve specific molar ratios for enhanced biocompatibility and biomimicry, combined with a biohybrid composite using natural or synthetic polymers like collagen for improved bone tissue integration.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Reliability

If stoichiometric hydroxyapatite is used as bone substitute, then material stability is maintained, but reabsorbability and osteogenesis are insufficient leading to slow bone integration

Engineering Contradiction:
ImprovereabsorbabilityVSAvoidmaterial stability
Core Design Contradiction:
ReliabilityVSStability of the object's composition

Solution Approach 1:

The patent applies parameter changes by substituting ions in the hydroxyapatite crystal structure with different elements (Sr, Si, Mg, CO3) to modify its chemical composition and physical properties. This enables the material to achieve both improved reabsorbability and osteogenesis while maintaining sufficient structural stability for bone substitution applications

Inventive Principle:
Principle #35Parameter changes

2Reliability

If stoichiometric hydroxyapatite is used as bone substitute, then material simplicity is maintained, but osteoblast activation is insufficient leading to slow bone regeneration

Engineering Contradiction:
Improveosteoblast activationVSAvoidmaterial complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent employs composite materials by creating multi-substituted hydroxyapatite containing multiple ion types (Sr2+, SiO4 4-, Mg2+, CO3 2-) within the hydroxyapatite structure. This composite approach at the atomic level provides synergistic effects that enhance osteoblast activation and bone regeneration while maintaining a single-phase material structure

Inventive Principle:
Principle #40Composite materials

3Productivity

If multi-substituted hydroxyapatite is developed to improve biocompatibility, then bone integration speed is enhanced, but manufacturing complexity increases

Engineering Contradiction:
Improvebone integration speedVSAvoidmanufacturing complexity
Core Design Contradiction:
ProductivityVSEase of manufacture

Solution Approach 1:

The patent applies preliminary action by pre-calculating and optimizing the molar ratios of substituting ions before synthesis. The specific molar ratios (Sr/Ca: 0.01-0.50, Si/PO4: 0.01-0.10, Mg/Ca: 0.01-0.20, CO3/PO4: 0.05-0.30) are determined in advance to achieve the desired biological performance, simplifying the manufacturing process by eliminating the need for iterative optimization

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The multi-substituted hydroxyapatite and biohybrid composite demonstrate enhanced reabsorbability, osteogenesis, and structural similarity to natural bone, facilitating faster bone remodeling and integration, thus serving as an effective and biocompatible bone substitute.

Implementation Method 1

hydroxyapatite multi-substituted with physiologically compatible ion species... Sr2+, and optionally silicate (SiO4 4-) and/or carbonate (CO3 2-) ions

Methodology Applied
Scientific EffectIonic substitution: Ion Exchange

Data Source

PatentEP1948561B1A plurisubstituted hydroxyapatite and the composite thereof with a natural and/or synthetic polymer, their preparation and uses thereof
Publication Date: 2016.09.07 FIN CERAMICA FAENZA
  • EP1948561B1 patent drawingFigure 1
  • EP1948561B1 patent drawingFigure 2
  • EP1948561B1 patent drawingFigure 3

AI summary

The present invention relates to a hydroxyapatite multi-substituted with, physiologically compatible ion species and to its biohybrid composite with a natural and/or synthetic polymer, which are useful in the preparation of a biomimetic bone substitute for treat¬ ing bone tissue defects. Furthermore, the present invention relates to a method for their preparation and uses .