Multi-Layer Nicotine Composition for Fast and Extended Release

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Existing nicotine delivery methods, such as lozenges and tablets, lack alternatives for providing a modified release profile and diverse organoleptic properties for therapeutic purposes.

Innovation Solution

A multi-layered nicotine-containing pharmaceutical composition comprising a core formulation surrounded by one or more layers with different organoleptic properties, including formulations with fast and extended release profiles, such as dissolvable, meltable, pastille, and chewable layers, to provide a unique delivery experience.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Adaptability or versatility

If a single formulation is used in nicotine delivery products, then the product structure is simple, but the release profile and organoleptic properties are limited

Engineering Contradiction:
Improverelease profile and organoleptic propertiesVSAvoidproduct structure
Core Design Contradiction:
Adaptability or versatilityVSDevice complexity

Solution Approach 1:

The nicotine delivery product is divided into multiple distinct formulations (first formulation and second formulation) with different properties. Each formulation can provide different release profiles (fast-release vs. extended-release) and organoleptic characteristics, allowing the product to offer versatile delivery options without requiring multiple separate products

Inventive Principle:
Principle #1Segmentation

Solution Approach 2:

One formulation is placed within or adjacent to another formulation in a multi-layered structure. The first formulation and second formulation are positioned in spatial relationship (e.g., core and coating, or adjacent layers) to enable simultaneous or sequential delivery of nicotine with different release profiles and sensory properties from a single integrated product

Inventive Principle:
Principle #7Nested doll (Nesting)

2Speed

If fast-release formulation is used, then immediate nicotine delivery is achieved, but duration of action is limited

Engineering Contradiction:
Improvenicotine release speedVSAvoidduration of nicotine delivery
Core Design Contradiction:
SpeedVSDuration of action of moving object

Solution Approach 1:

The invention combines fast-release formulation and extended-release formulation into a single nicotine delivery product. The fast-release component provides immediate nicotine delivery to satisfy acute cravings, while the extended-release component simultaneously provides prolonged nicotine supply to maintain therapeutic levels over time, thus merging the benefits of both release profiles in one product

Inventive Principle:
Principle #5Merging (Combining)

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The multi-layered composition offers a tailored release profile and varied sensory experience, enhancing therapeutic efficacy and user satisfaction.

Implementation Method 1

the nicotinic compound-containing pharmaceutical composition comprises a nicotinic compound sorbed onto a porous particulate carrier

Methodology Applied
Scientific EffectSorption: Sorption

Data Source

PatentEP3735972B1Multi-layer nicotine-containing pharmaceutical composition
Publication Date: 2025.11.19 MODORAL BRANDS INC

AI summary

The invention provides a multi-layered pharmaceutical composition comprising two or more formulations with varying properties. In some embodiments, the pharmaceutical compositions provide combinations of different organoleptic properties within the same product. In certain embodiment, these combinations allow for a modified release profile of active ingredients as the user enjoys the pharmaceutical composition. The invention further provides methods for making and using the pharmaceutical composition.