Nitrogen-Containing Surfactants for Glyphosate Formulations

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current surfactants used in agricultural formulations, such as tallowamine ethoxylate, enhance pesticide efficacy but have unfavorable aquatic toxicity and eye irritation profiles, and there is a need for surfactants that can improve bioefficacy while reducing toxicity and irritation without compromising stability in various glyphosate formulations.

Innovation Solution

The use of nitrogen-containing surfactants with specific structures, including alkyl imino dipropionates and amine oxides, which are compatible in high load ammonium and potassium glyphosate formulations, and can enhance the efficacy of agricultural formulations without the need for additional compatibility agents.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If traditional surfactants like tallowamine ethoxylate are used to enhance pesticide efficacy, then bioefficacy is improved, but aquatic toxicity and eye irritation increase

Engineering Contradiction:
ImprovebioefficacyVSAvoidaquatic toxicity and eye irritation
Core Design Contradiction:
ProductivityVSObject-affected harmful factors

Solution Approach 1:

The patent changes the chemical structure parameters of the surfactant by introducing nitrogen-containing functional groups (amino, amido, or amine oxide groups) at specific positions in the molecular structure. This structural modification allows the surfactant to maintain effective bioefficacy while reducing aquatic toxicity and eye irritation compared to traditional surfactants like tallowamine ethoxylate

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent creates composite surfactant molecules combining hydrophobic alkyl groups (C12-C22) with hydrophilic nitrogen-containing functional groups (amino, amido, or amine oxide). This composite structure enables the surfactant to achieve both effective bioefficacy enhancement and reduced toxicity profiles by balancing lipophilicity and hydrophilicity in a single molecular architecture

Inventive Principle:
Principle #40Composite materials

2Object-affected harmful factors

If surfactants with better aquatic toxicity and eye irritation profiles are used, then environmental safety is improved, but bioefficacy enhancement decreases

Engineering Contradiction:
Improveaquatic toxicity and eye irritationVSAvoidbioefficacy
Core Design Contradiction:
Object-affected harmful factorsVSProductivity

Solution Approach 1:

The patent optimizes the nitrogen-containing functional group parameters (amino, amido, or amine oxide) and their positions in the molecular structure to achieve the right balance between environmental safety and bioefficacy. The specific structural parameters (R groups, m, n, p, q values) are tuned to maintain surfactant effectiveness while ensuring reduced toxicity

Inventive Principle:
Principle #35Parameter changes

3Object-affected harmful factors

If new surfactant structures are developed to replace traditional surfactants, then toxicity profiles are improved, but formulation stability may be compromised

Engineering Contradiction:
Improvetoxicity profilesVSAvoidformulation stability
Core Design Contradiction:
Object-affected harmful factorsVSStability of the object's composition

Solution Approach 1:

The patent carefully adjusts the chemical parameters of the new surfactant structure, including the alkyl chain length (C12-C22), the type of nitrogen-containing group (amino, amido, or amine oxide), and the ethoxylate chain length (m and n values). These parameter optimizations ensure that the new surfactant maintains compatibility and stability in various agricultural formulations while achieving improved toxicity profiles

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent introduces specific local functional groups (amino, amido, or amine oxide) at defined positions in the surfactant molecule while maintaining the overall surfactant architecture. This localized modification allows the new surfactant to achieve reduced toxicity while preserving the structural features necessary for formulation stability

Inventive Principle:
Principle #3Local quality

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

These surfactants demonstrate improved bioefficacy and stability in concentrated glyphosate formulations, reducing aquatic toxicity and eye irritation while maintaining or exceeding the efficacy of traditional surfactants, even at lower concentrations, and are compatible in various glyphosate salt forms.

Implementation Method 1

The bioefficacy of pesticides is known to be enhanced by the addition of appropriate surfactants, or adjuvants

Methodology Applied
Scientific EffectSurface tension reduction: Surface Tension

Data Source

PatentEP4029374A1Nitrogen containing surfactants for agricultural use
Publication Date: 2022.07.20 AKZO NOBEL CHEMICALS INTERNATIONAL BV
  • EP4029374A1 patent drawingFigure 1~2
  • EP4029374A1 patent drawingFigure 3~4
  • EP4029374A1 patent drawingFigure 5~6

AI summary

An agricultural formulation comprises: at least one agricultural active; and an alkyl imino dipropionate having the formula: wherein R is a C6 - C24, linear or branched, alkyl group, and wherein each M is independently a cation chosen from Mg2+, Ca2+, NH4 +, K+, and Na+, and wherein the formulation is free of an alkylamine and/or derivative thereof if R is lauryl.