Omega-3 Fatty Acid Amino Acid Salt Tablets

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Solution Overview

Problem

Current omega-3 fatty acid products, particularly in solid forms, face challenges such as low bioavailability, sensitivity to oxidation, high costs, and low concentration, leading to the need for frequent and large doses to achieve recommended daily intake.

Innovation Solution

Development of tablets comprising omega-3 fatty acid amino acid salts with reduced content of binders and structure-forming substances, such as polyvinylpyrrolidone, starch, and calcium phosphate, allowing for high omega-3 fatty acid content and improved bioavailability without the need for additional auxiliaries.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Stability of the object's composition

If omega-3 fatty acid products are formulated with high content of binders and structure-forming substances to ensure tablet stability, then tablet structural integrity is improved, but omega-3 fatty acid content and bioavailability are reduced

Engineering Contradiction:
Improvetablet structural integrityVSAvoidomega-3 fatty acid content
Core Design Contradiction:
Stability of the object's compositionVSQuantity of substance

Solution Approach 1:

The patent changes the concentration parameter by reducing binder content from conventional levels (typically 30-50% in solid formulations) to minimal or zero levels, while maintaining tablet integrity through the unique properties of omega-3 fatty acid amino acid salts that require no additional binders or structure-forming substances

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent extracts and removes binders and structure-forming substances from the formulation, achieving a pure omega-3 fatty acid amino acid salt composition without conventional tablet excipients, thereby maximizing omega-3 content while maintaining structural integrity

Inventive Principle:
Principle #2Taking out (Extraction)

2Ease of manufacture

If conventional solid formulations use multiple auxiliaries and binders to ensure manufacturability, then ease of manufacture is improved, but product purity and omega-3 concentration are reduced

Engineering Contradiction:
Improvetablet manufacturabilityVSAvoidomega-3 fatty acid concentration
Core Design Contradiction:
Ease of manufactureVSQuantity of substance

Solution Approach 1:

The omega-3 fatty acid amino acid salt serves its own structural and binding functions, eliminating the need for separate binders and structure-forming substances, thereby achieving both high concentration and ease of manufacture through a self-sufficient formulation

Inventive Principle:
Principle #25Self-service

Solution Approach 2:

The patent changes the formulation composition parameter by eliminating auxiliary substances entirely, relying solely on the omega-3 fatty acid amino acid salt which inherently possesses all necessary properties for tablet formation without additional manufacturability aids

Inventive Principle:
Principle #35Parameter changes

3Loss of substance

If low concentration formulations are used to reduce costs, then manufacturing cost is reduced, but daily intake requirements necessitate large doses and frequent administration

Engineering Contradiction:
Improvemanufacturing costVSAvoiddaily intake amount
Core Design Contradiction:
Loss of substanceVSQuantity of substance

Solution Approach 1:

The patent changes the concentration parameter by producing ultra-pure omega-3 fatty acid amino acid salts with minimal excipients, enabling high-dose delivery in small tablet quantities, thereby reducing both manufacturing cost per effective dose and the physical burden of administration on consumers

Inventive Principle:
Principle #35Parameter changes

4Reliability

If conventional formulations use animal-derived gelatine or plant-based capsules, then encapsulation and protection are improved, but consumer acceptance is reduced due to religious or dietary restrictions

Engineering Contradiction:
Improveencapsulation protectionVSAvoidconsumer acceptance
Core Design Contradiction:
ReliabilityVSAdaptability or versatility

Solution Approach 1:

The patent extracts and eliminates animal-derived gelatine and plant-based capsule materials from the formulation, replacing them with a pure omega-3 fatty acid amino acid salt tablet that requires no controversial encapsulation materials, thereby achieving universal consumer acceptance while maintaining product integrity

Inventive Principle:
Principle #2Taking out (Extraction)

Solution Approach 2:

The patent replaces the conventional capsule encapsulation concept with a direct tablet formulation that inherently provides the same protective and delivery functions without using gelatine or plant-based materials, offering a universally acceptable alternative

Inventive Principle:
Principle #26Copying

Data Source

PatentUS12115260B2Tablets with high active ingredient content of omega-3 fatty acid amino acid salts
Publication Date: 2024.10.15 EVONIK OPERATIONS GMBH

AI summary

The present invention relates to a tablet comprising one or more omega-3 fatty acid amino acid salt(s), a method for preparing a tablet according to the invention and the use of a tablet according to the invention as a food supplement or as a pharmaceutical product.