Optimized Transcription Terminator Sequences for Recombinant Protein Yield

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Solution Overview

Problem

Current recombinant protein expression systems face challenges in achieving high yield and efficiency due to antagonistic relationships between high expression rates and cell viability, with inefficient transcriptional termination leading to metabolic burdens and unwanted protein expression.

Innovation Solution

Incorporation of polynucleotides with optimized transcription termination signals, specifically hairpin structures with high G/C content and complementary sequences, to enhance termination efficiency and control expression rates.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Productivity

If high expression rates are used to increase recombinant protein yield, then productivity is improved, but cell viability deteriorates due to metabolic burden

Engineering Contradiction:
Improverecombinant protein yieldVSAvoidcell viability
Core Design Contradiction:
ProductivityVSReliability

Solution Approach 1:

The patent optimizes transcription termination efficiency by modifying terminator sequence parameters (G/C content, hairpin structure, length) to control the duration and intensity of transcription. This regulates gene expression levels to reduce metabolic burden on cells while maintaining adequate protein production, thus resolving the contradiction between productivity and cell viability

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent employs inducible promoter systems that allow periodic control of gene expression. Transcription can be activated only when needed and terminated efficiently when not required, enabling cells to alternate between production mode and recovery mode, thereby maintaining viability while achieving high overall productivity

Inventive Principle:
Principle #19Periodic action

2Productivity

If transcription termination efficiency is low, then read-through transcription occurs producing lengthy mRNAs, but this increases metabolic burden and causes unwanted protein expression

Engineering Contradiction:
Improvetranscription efficiencyVSAvoidmetabolic burden
Core Design Contradiction:
ProductivityVSObject-generated harmful factors

Solution Approach 1:

The patent systematically optimizes terminator sequence parameters including increasing G/C content to 70-80%, adjusting hairpin stem length to 10-15 base pairs, and optimizing loop structure to achieve termination efficiency above 90%. These parameter changes ensure efficient transcription termination that prevents read-through transcription and eliminates the harmful metabolic burden while maintaining high transcription efficiency

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent utilizes the physical-chemical properties of RNA secondary structures (hairpin formations) to create a mechanical barrier that physically blocks the RNA polymerase. The optimized hairpin structure acts like a physical stop mechanism, using base-pairing energy and structural geometry to force termination, thereby preventing harmful read-through transcription

Inventive Principle:
Principle #29Pneumatics and hydraulics

3Reliability

If termination signals are optimized with high G/C content and stable hairpin structures, then termination efficiency is improved, but the complexity of the terminator sequence increases

Engineering Contradiction:
Improvetermination efficiencyVSAvoidterminator sequence complexity
Core Design Contradiction:
ReliabilityVSDevice complexity

Solution Approach 1:

The patent establishes specific parameter ranges for terminator sequences: G/C content of 70-80%, hairpin stem length of 10-15 base pairs, and loop length of 4-8 nucleotides. These standardized parameters provide a systematic approach to designing efficient terminators without arbitrary complexity, making the design process more predictable and manageable

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent applies different structural requirements to different regions of the terminator sequence. The stem region requires high G/C content for stability, the loop region has specific length constraints for proper folding, and the overall structure follows defined geometric parameters. This localized optimization achieves high termination efficiency while maintaining structured simplicity

Inventive Principle:
Principle #3Local quality

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The use of optimized termination signals significantly increases termination efficiency, reducing metabolic burdens and improving recombinant protein production while maintaining cell viability.

Implementation Method 1

a hairpin structure comprising a stem of at least 12 internal base pairs... Z is a nucleotide sequence with at least 70% complementarity to Y, the complementary nucleotides of Z being base paired with the nucleotides of Y

Methodology Applied
Scientific EffectBase pairing: Chemical Bonding

Implementation Method 2

the enzyme moves along the template, incorporates nucleotides one by one and produces the desired RNA chain

Methodology Applied
Scientific EffectNucleotide incorporation: Chemical Bonding

Data Source

PatentEP2714913B1Transcription terminator sequences
Publication Date: 2018.04.25 SANDOZ LTD
  • EP2714913B1 patent drawingFigure 1
  • EP2714913B1 patent drawingFigure 2a~2b
  • EP2714913B1 patent drawingFigure 3a~4b

AI summary

The present invention provides new transcription termination signal sequences, especially a polynucleotide comprising at least two consecutive transcription termination signals, characterized in that said consecutive transcription termination signals comprise at least a first and a second transcription termination signal that are at most 1000 nucleotides apart, and at least one of the termination signal has or encodes a RNA hairpin structure.