Optogenetic Action Potential Interception via Light-Activated Protein Systems

Resolve Bottlenecks,
Find Innovative Solutions
Generate Solutions

Solution Overview

Problem

Current optogenetic tools face limitations in effectively inhibiting and intercepting action potentials in target cells due to weak photocurrents and reduced specificity, particularly in optogenetic electrical inhibition and excitation, which affects the precision and specificity of neural modulation.

Innovation Solution

The development of systems and methods utilizing light-activated proteins, such as eArch3.0 and ASIC2a, which are delivered to target cells via nucleic acids and expression systems, allowing for optogenetic modulation of action potentials, including inhibition and interception, using light-activated proteins that facilitate ion passage across cell membranes and response proteins that enhance ion flow.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Power

If existing ion pump proteins are used for optogenetic inhibition, then temporal precision is achieved, but photocurrent strength is weak and input resistance changes are insufficient

Engineering Contradiction:
Improvephotocurrent strengthVSAvoidinhibition effectiveness
Core Design Contradiction:
PowerVSReliability

Solution Approach 1:

The patent combines a light-activated protein (e.g., eArch3.0 proton pump) with a response protein (ASIC2a acid-sensitive ion channel) to create a two-component system. The light-activated protein generates acidification that activates the response protein, which then opens ion channels to produce strong inward currents. This merging of components resolves the contradiction by transforming weak photocurrents into strong, reliable inhibition currents while maintaining temporal precision.

Inventive Principle:
Principle #5Merging (Combining)

2Measurement precision

If light-activated proteins are used for optogenetic excitation, then temporal precision is achieved, but specificity is reduced due to retrograde propagating action potentials

Engineering Contradiction:
ImprovespecificityVSAvoidretrograde action potential propagation
Core Design Contradiction:
Measurement precisionVSObject-generated harmful factors

Solution Approach 1:

The patent extracts and targets action potentials at specific locations (such as axon initial segments or synapses) using spatially selective light stimulation. By applying light only to specific regions where action potentials are generated or transmitted, the system can intercept and inhibit these potentials before they propagate retrogradely to the cell body, thereby maintaining specificity while preventing harmful retrograde propagation.

Inventive Principle:
Principle #2Taking out (Extraction)

3Manufacturing precision

If existing optogenetic tools are used, then cell-type resolution is maintained, but functional precision is insufficient for intercepting action potentials

Engineering Contradiction:
Improvefunctional precisionVSAvoidsystem complexity
Core Design Contradiction:
Manufacturing precisionVSDevice complexity

Solution Approach 1:

The patent segments the optogenetic system into distinct functional components: light-activated proteins for local acidification, response proteins for ion channel activation, and delivery mechanisms for targeted expression. This segmentation allows each component to be optimized independently for its specific function while working together to achieve precise action potential interception, thereby improving functional precision without excessive overall complexity.

Inventive Principle:
Principle #1Segmentation

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

These systems enable precise modulation of action potentials, improving the specificity and effectiveness of optogenetic interventions in neural applications, such as treating neurological and psychiatric conditions by effectively inhibiting and intercepting action potentials.

Implementation Method 1

light-activated proteins, such as eArch3.0 and ASIC2a, which are delivered to target cells via nucleic acids and expression systems, allowing for optogenetic modulation of action potentials

Methodology Applied
Scientific EffectPhotoelectric Effect: Photoelectric Effect

Data Source

PatentEP2991491B1Devices, systems and methods for optogenetic modulation of action potentials in target cells
Publication Date: 2019.12.25 THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIV
  • EP2991491B1 patent drawingFigure 1
  • EP2991491B1 patent drawingFigure 2
  • EP2991491B1 patent drawingFigure 3A~3B

AI summary

Aspects of the disclosure include devices, systems and methods for optogenetic modulation of action potentials in target cells. The subject devices include light-generating devices, control devices, and delivery devices for delivering vectors to target cells. The subject systems include light-activated proteins, response proteins, nucleic acids comprising nucleotide sequences encoding these proteins, as well as expression systems that facilitate expression of these proteins in target cells. Also provided are methods of using the subject devices and systems to optogenetically inhibit and intercept action potentials in target cells, e.g., to treat a neurological or psychiatric condition in a human or non-human animal subject.