Oral Therapeutic Composition for Dry Eye Syndrome

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Solution Overview

Problem

Current treatments for dry eye syndrome and vitreous opacities, such as artificial tears and surgical procedures, provide only temporary relief and are not effective in addressing the underlying issues of tear film instability and ocular surface disease.

Innovation Solution

An orally administered composition comprising a mixture of water-soluble and water-insoluble antioxidants, essential fatty acids, glycoprotein complex, phospholipids, phytosterols, curcuminoids, and micronutrient cofactors like vitamin B6 and copper, which synergistically replenishes the tear film layers, reduces inflammation, and stabilizes the tear film.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Duration of action of moving object

If artificial tears are administered to treat dry eye syndrome, then temporary rehydration of the eyes is achieved, but relief is short-lived and frequent dosing is necessary

Engineering Contradiction:
Improveduration of reliefVSAvoidfrequency of dosing
Core Design Contradiction:
Duration of action of moving objectVSProductivity

Solution Approach 1:

The patent applies preliminary action by administering oral supplements (omega-3 fatty acids, antioxidants, vitamins) before the actual tear production issue occurs. These supplements prepare the body's systems in advance to naturally produce better-quality tears and reduce inflammation, thereby extending the duration of relief and reducing the need for frequent artificial tear dosing.

Inventive Principle:
Principle #10Preliminary action

Solution Approach 2:

The patent enables self-service by stimulating the body's own natural tear production mechanisms through oral supplementation. Instead of relying continuously on external artificial tears, the composition helps the patient's lacrimal glands and ocular surface cells regenerate and produce their own protective tear film, reducing dependence on frequent external interventions.

Inventive Principle:
Principle #25Self-service

2Reliability

If artificial tears are used to treat dry eye syndrome, then temporary rehydration is achieved, but contra-indications and incompatibility with soft contact lenses occur

Engineering Contradiction:
Improvecompatibility with contact lensesVSAvoidcontra-indications
Core Design Contradiction:
ReliabilityVSObject-affected harmful factors

Solution Approach 1:

The patent enables self-service by stimulating the body's own natural tear production mechanisms through oral supplementation. Instead of relying continuously on external artificial tears, the composition helps the patient's lacrimal glands and ocular surface cells regenerate and produce their own protective tear film, reducing dependence on frequent external interventions.

Inventive Principle:
Principle #25Self-service

3Reliability

If current medications are administered for xerophthalmia syndrome, then treatment is attempted, but only limited results are achieved

Engineering Contradiction:
Improveeffectiveness of treatmentVSAvoidclinical outcome
Core Design Contradiction:
ReliabilityVSProductivity

Solution Approach 1:

The patent applies composite materials by combining multiple active ingredients in a synergistic formulation: omega-3 fatty acids (for tear film stability and anti-inflammatory effects), antioxidants like vitamins C and E (for protecting ocular cells from oxidative damage), and other supportive nutrients. This multi-component composite approach addresses multiple aspects of dry eye pathophysiology simultaneously, achieving better clinical outcomes than single-agent medications.

Inventive Principle:
Principle #40Composite materials

Solution Approach 2:

The patent converts harmful oxidative stress and inflammation into beneficial effects by using antioxidants and anti-inflammatory omega-3 fatty acids to neutralize free radicals and reduce inflammatory mediators. The composition transforms the harmful oxidative environment that contributes to dry eye disease into a protective antioxidant-rich environment that promotes ocular surface healing and tear film stability.

Inventive Principle:
Principle #22Blessing in disguise (Convert harm into benefit)

Data Source

PatentUS7638142B2Therapeutic composition for the treatment of dry eye syndrome
Publication Date: 2009.12.29 VITAMIN SCIENCE LLC

AI summary

A composition and method for treating dry-eye syndrome and symptoms of vitreous opacities in a host comprising the oral administration of a composition which contains a pharmacologically effective amount of essential fatty acids, polar phospholipids, vitamins, minerals and dietary supplements.