Oral Paste Carrier for Canker Sore Treatment

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Solution Overview

Problem

Current canker sore treatments either lack an anti-inflammatory component or are ineffective in maintaining a local anesthetic presence, leading to prolonged healing times and discomfort due to quick dissipation in a saliva-rich environment.

Innovation Solution

A topical composition combining 10-30% benzocaine as an anesthetic with 0.5-2% hydrocortisone, carried by a paste formulation including sodium carboxymethylcellulose, gelatin, citrus, pectin, petrolatum, and titanium dioxide, which resists washing away and provides sustained delivery.

Engineering Contradictions & Design Principles

VSEngineering Contradiction Analysis

1Duration of action of moving object

If a gel-based carrier is used to deliver anesthetic and anti-inflammatory substances, then the composition can be applied topically to the canker sore, but the carrier quickly dries up and washes away with saliva, reducing treatment effectiveness

Engineering Contradiction:
Improveduration of treatment effectivenessVSAvoidstability of carrier in saliva environment
Core Design Contradiction:
Duration of action of moving objectVSStability of the object's composition

Solution Approach 1:

The patent changes the physical state of the carrier from gel to paste, and adjusts the concentration of hydrophilic and lipophilic components to create a balanced formulation that resists both drying and washing away. The paste form maintains moisture while the specific composition ratio (40-60% hydrophilic, 40-60% lipophilic) provides stability in the saliva environment.

Inventive Principle:
Principle #35Parameter changes

Solution Approach 2:

The patent uses a composite carrier system combining multiple ingredients with different properties: hydrophilic agents (sodium carboxymethylcellulose, gelatin, pectin) for water retention, lipophilic agents (petrolatum, titanium dioxide) for water resistance, and adhesive agents (vanillin) for bonding to the sore. This composite approach creates a carrier that simultaneously resists drying, washing away, and detachment.

Inventive Principle:
Principle #40Composite materials

2Object-affected harmful factors

If only anesthetic substances are used to treat canker sores, then pain is relieved, but inflammation is not addressed, prolonging healing time

Engineering Contradiction:
Improvepain reliefVSAvoidhealing duration
Core Design Contradiction:
Object-affected harmful factorsVSLoss of time

Solution Approach 1:

The patent combines two previously separate treatment approaches (anesthetic-only and anti-inflammatory-only) into a single dual-action composition. The formulation includes both benzocaine (anesthetic) and hydrocortisone (anti-inflammatory) in specific concentrations (10-30% and 0.5-2% respectively), allowing simultaneous pain relief and inflammation reduction to accelerate healing.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The patent creates a multi-functional treatment composition that performs multiple functions: analgesic (benzocaine), anti-inflammatory (hydrocortisone), and carrier/stabilizer (paste formulation with hydrophilic and lipophilic agents). This universal composition addresses both pain and inflammation while maintaining stability in the oral environment.

Inventive Principle:
Principle #6Universality (Multi-functionality)

3Object-affected harmful factors

If only anti-inflammatory substances are used to treat canker sores, then inflammation is reduced, but application is painful and effects are delayed without local anesthetic

Engineering Contradiction:
Improveinflammation reductionVSAvoidease of application
Core Design Contradiction:
Object-affected harmful factorsVSEase of operation

Solution Approach 1:

The patent combines anti-inflammatory hydrocortisone (0.5-2%) with local anesthetic benzocaine (10-30%) in a single formulation. This allows the composition to reduce inflammation while simultaneously numbing the area to eliminate application pain, making the treatment both effective and comfortable.

Inventive Principle:
Principle #5Merging (Combining)

Solution Approach 2:

The anesthetic component acts preliminarily by numbing the canker sore area before the anti-inflammatory component takes effect. This preliminary analgesic action makes the application of the anti-inflammatory substance painless and allows the inflammation-reducing effects to develop without patient discomfort.

Inventive Principle:
Principle #10Preliminary action

Applied Scientific Principles

This section explains which scientific principles are used to turn an abstract innovation direction into a practical engineering solution.

Function Achieved in This Case

The composition significantly reduces pain and inflammation, shrinking lesions by half within 24 hours and shortening healing duration to 7-14 days, while maintaining adhesive properties to withstand saliva, allowing for effective treatment without frequent reapplication.

Implementation Method 1

a paste carrier to carry and apply the anesthetic substance and the anti-inflammatory substance directly to a canker sore

Methodology Applied
Scientific EffectAdhesion: Adhesive

Implementation Method 2

In order to resist quick drying and/or washing away from the canker sore site, the paste carrier may include sodium carboxymethylcellulose, gelatin, citrus, pectin, petrolatum, and titanium dioxide

Methodology Applied
Scientific EffectHydrophobicity: Hydrophobe

Data Source

PatentUS11622953B2Oral composition for the treatment of canker sores
Publication Date: 2023.04.11 VARANI ANTOINE

AI summary

A composition, and method for using the same, for treating a canker sore includes 10-30% of an ester local anesthetic, 0.5-2% of a corticosteroid, and a carrier for the ester local anesthetic and the corticosteroid. The carrier is formulated as a paste so as to be applied topically to the canker sore to deliver the ester local anesthetic and the corticosteroid simultaneously to the canker sore.